Muraglitazar

Muraglitazar

SCHEMBL676469

COc1ccc(OC(=O)N(CC(=O)O)Cc2ccc(OCCc3nc(-c4ccccc4)oc3C)cc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPARAPPARG

The experimentally established mechanism targets of Muraglitazar. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PPARA known ✓ Q07869 19/20 1.00
PPARG known ✓ P37231 17/20 1.00
CYP2C9 P11712 1/20 0.65
KCNH2 Q12809 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13722049 0.96 PPARA (0.93) PPARAPPARGCYP2C9KCNH2
SCHEMBL13718146 0.96 PPARA (0.93) PPARAPPARGCYP2C9KCNH2
SCHEMBL6073227 0.95 PPARA (0.90) PPARAPPARGCYP2C9KCNH2
SCHEMBL8215885 0.94 PPARA (0.88) PPARAPPARG
SCHEMBL6073514 0.94 PPARA (0.88) PPARAPPARGCYP2C9KCNH2
SCHEMBL13721992 0.93 PPARA (0.87) PPARAPPARGCYP2C9KCNH2
SCHEMBL13717685 0.93 PPARA (0.87) PPARAPPARGCYP2C9KCNH2
SCHEMBL13717584 0.93 PPARA (0.89) PPARAPPARGCYP2C9KCNH2
SCHEMBL13718351 0.93 PPARA (0.89) PPARAPPARGCYP2C9KCNH2
SCHEMBL13717851 0.93 PPARA (0.87) PPARAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1291 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137661-A1 PPAR-ALPHA/GAMMA AGONIST FOR USE IN THE TREATMENT OF LIVER FAILURE GENFIT (FR) 2026-05-21 US claimed
US-20260108482-A1 MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X4 AND RELATED PRODUCTS AND METHODS ESCIENT PHARMACEUTICALS INC (US) 2026-04-23 US claimed
EP-4725479-A1 PPAR AGONISTS FOR TREATMENT OF DISEASES ASSOCIATED WITH AATD Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2026-04-15 EP claimed
EP-3452041-B1 COMPOSITIONS AND METHODS FOR ADMINISTERING PPAR-GAMMA-AGONISTS, SURFACTANT PEPTIDES AND PHOSPHOLIPIDS LOS ANGELES BIOMEDICAL RES INST HARBOR UCLA MEDICAL CT (US) 2026-01-14 EP claimed
US-20250367217-A1 PHARMACEUTICAL COMPOSITIONS FOR COMBINATION THERAPY INTERCEPT PHARMACEUTICALS INC (US) 2025-12-04 US claimed
US-20250367216-A1 PHARMACEUTICAL COMPOSITIONS FOR COMBINATION THERAPY INTERCEPT PHARMACEUTICALS INC (US) 2025-12-04 US claimed
EP-4615433-A1 PPAR-ALPHA/GAMMA AGONIST FOR USE IN THE TREATMENT OF LIVER FAILURE Genfit (FR) 2025-09-17 EP claimed
EP-3787631-B1 MODULATORS OF ORPHAN NUCLEAR RECEPTORS FOR NASH AND OTHER METABOLIC DISORDERS UNIV EMORY (US) 2025-09-10 EP claimed
EP-4558622-A1 METHODS AND COMPOSITIONS FOR GENERATING HUMAN MIDBRAIN DOPAMINERGIC NEURONS FROM NEURAL PROGENITOR CELLS Trailhead Biosystems Inc. (US) 2025-05-28 EP claimed
US-20250082781-A1 METHODS OF LOWERING BLOOD GLUCOSE AND TREATING TYPE 2 DIABETES BY ACTIVATION OF PDE4D3 SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 2025-03-13 US claimed
WO-2016127019-A2 PHARMACEUTICAL COMPOSITIONS FOR COMBINATION THERAPY INTERCEPT PHARMACEUTICALS, INC. (US) 2016-08-11 WO claimed
US-20160128994-A1 PPAR GAMMA MODULATORS FOR TREATING CYSTIC DISEASES INDIANA UNIVERSITY RESEARCH & TECHNOLOGY CORPORATION (US) 2016-05-12 US claimed
EP-3003303-A1 PPAR GAMMA MODULATORS FOR TREATING CYSTIC DISEASES Indiana University Research And Technology Corporation (US) 2016-04-13 EP claimed
WO-2014197820-A1 PPAR GAMMA MODULATORS FOR TREATING CYSTIC DISEASES INDIANA UNIVERSITY RESEARCH & TECHNOLOGY CORPORATION (US) 2014-12-11 WO claimed
EP-2253325-A1 AGENT FOR ENHANCING CORNEAL EPITHELIAL BARRIER FUNCTION Santen Pharmaceutical Co., Ltd (JP) 2010-11-24 EP claimed
US-7348329-B2 Therapeutic agent for keratoconjunctival disorder SANTEN PHARMACEUTICAL CO., LTD. (JP) 2008-03-25 US claimed
US-20070093514-A1 Therapeutic agent for keratoconjunctival disorder SANTEN PHARMACEUTICAL CO., LTD. (JP) 2007-04-26 US claimed
US-20060177444-A1 Concomitant drug as therapeutic agent for inflammatory bowel disease EISAI R&D MANAGEMENT CO., LTD. (JP) 2006-08-10 US claimed
EP-1681054-A1 THERAPEUTIC AGENT FOR KERATOCONJUNCTIVA DISORDER SANTEN PHARMACEUTICAL CO., LTD. (JP) 2006-07-19 EP claimed
EP-1607103-A1 CONCOMITANT DRUG AS THERAPEUTIC AGENT FOR INFLAMMATORY BOWEL DISEASE Eisai Co., Ltd. (JP) 2005-12-21 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260137661-A1 PPAR-ALPHA/GAMMA AGONIST FOR USE IN THE TREATMENT OF LIVER FAILURE PPARA, PPARD, PPARG PPARA 1/4885PPARG 3/4885CYP2C9 2389/4885
US-20250082781-A1 METHODS OF LOWERING BLOOD GLUCOSE AND TREATING TYPE 2 DIABETES BY ACTIVATION OF PDE4D3 PDE4D, PDE4A, PDE4B PPARA 210/4885PPARG 129/4885CYP2C9 3760/4885
US-20250367216-A1 PHARMACEUTICAL COMPOSITIONS FOR COMBINATION THERAPY PPARD, NR1H4, PPARG PPARA 4/4885PPARG 3/4885CYP2C9 402/4885
US-20260108482-A1 MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X4 AND RELATED PRODUCTS AND METHODS MRGPRX4, MRGPRX1, MRGPRX2 PPARA 1336/4885PPARG 467/4885CYP2C9 1471/4885
US-20060177444-A1 Concomitant drug as therapeutic agent for inflammatory bowel disease PPARG, PPARA, NR3C1 PPARA 2/4885PPARG 1/4885CYP2C9 2362/4885
US-20250367217-A1 PHARMACEUTICAL COMPOSITIONS FOR COMBINATION THERAPY PPARD, NR1H4, PPARG PPARA 4/4885PPARG 3/4885CYP2C9 402/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.