SCHEMBL6767923

SCHEMBL6767923

O=C(O)c1nnn[nH]1.[NaH].[NaH]

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.32
CGAS Q8N884 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1238342 0.97
Fluoride SCHEMBL30940539 0.95
SCHEMBL6316087 0.95 LMNA (0.32) LMNACGAS
SCHEMBL29576729 0.82 ADORA3 (0.30)
Tetrazole SCHEMBL30486918 0.80 HAO1 (0.31) CGAS
Tetrazole SCHEMBL29908245 0.80 CGAS (0.31) CGAS
SCHEMBL8099243 0.79
SCHEMBL10854768 0.78
SCHEMBL361611 0.75
SCHEMBL968348 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0670835-B1 PROCESS FOR PREPARING BENZOPYRAN COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 2003-03-12 EP claimed
US-5596103-A Process for preparing benzopyran compounds SMITHKLINE BEECHAM PLC (GB) 1997-01-21 US claimed
US-5587483-A Process for preparing tetrazol-5-yl substituted benzopyran compounds SMITHKLINE BEECHAM PLC (GB) 1996-12-24 US claimed
EP-0670835-A1 PROCESS FOR PREPARING BENZOPYRAN COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 1995-09-13 EP claimed
CN-1107153-A Process SMITHKLINE BEECHAM PLC (GB) 1995-08-23 CN claimed
WO-1994012492-A1 PROCESS FOR PREPARING BENZOPYRAN COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 1994-06-09 WO claimed
JP-5005918-A None JP disclosed
JP-2004035570-A METHOD FOR PRODUCING INTERMEDIATE FOR SYNTHESIZING PRECURSOR OF BENZOPYRAN COMPOUND SMITHKLINE BEECHAM PLC 2004-02-05 JP disclosed
EP-0670835-B1 PROCESS FOR PREPARING BENZOPYRAN COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 2003-03-12 EP disclosed
CN-1049657-C Process SMITHKLINE BEECHAM PLC (GB) 2000-02-23 CN disclosed
US-5777128-A Process for preparing benzopyran compounds SMITHKLINE BEECHAM P.L.C. (GB) 1998-07-07 US disclosed
US-5616721-A Process for preparing benzopyran compounds SMITHKLINE BEECHAM PLC (GB) 1997-04-01 US disclosed
EP-0760816-A1 PROCESS FOR PREPARING BENZOPYRAN COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 1997-03-12 EP disclosed
EP-0670835-A1 PROCESS FOR PREPARING BENZOPYRAN COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 1995-09-13 EP disclosed
CN-1107153-A Process SMITHKLINE BEECHAM PLC (GB) 1995-08-23 CN disclosed
WO-1994018178-A1 PROCESS FOR PREPARING TETRAZOLE-5-CARBOXYLIC ACID DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 1994-08-18 WO disclosed
WO-1994012492-A1 PROCESS FOR PREPARING BENZOPYRAN COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 1994-06-09 WO disclosed
JP-H055918-A NONLINEAR OPTICAL MATERIAL MATSUSHITA ELECTRIC IND CO LTD 1993-01-14 JP disclosed
CN-1035664-A NEW CHEMICAL PROCESS MAY & BAKER LTD (GB) 1989-09-20 CN disclosed
EP-0323885-A1 New chemical process MAY & BAKER LIMITED (GB) 1989-07-12 EP disclosed