SCHEMBL6770698

SCHEMBL6770698

CCOC(=O)C(CCn1cnc2c(Cl)nc(N)nc21)(C(=O)O)C(=O)OCC

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 17/20 0.48
HSP90AA1 P07900 16/20 0.48
CYP2C19 P33261 1/20 0.44
HSP90B1 P14625 1/20 0.44
TRAP1 Q12931 1/20 0.44
HDAC6 Q9UBN7 2/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6153979 0.95 HSP90AB1 (0.50) HSP90AB1HSP90AA1CYP2C19HSP90B1TRAP1
SCHEMBL7813344 0.83 CYP2C19 (0.46) HSP90AB1HSP90AA1CYP2C19HDAC1
SCHEMBL14227939 0.80 HSP90AB1 (0.43) HSP90AB1HSP90AA1CYP2C19HSP90B1TRAP1
SCHEMBL10521672 0.78 HSP90AB1 (0.39) HSP90AB1HSP90AA1HSP90B1TRAP1HDAC6
SCHEMBL28451668 0.78 HSP90AB1 (0.49) HSP90AB1HSP90AA1CYP2C19HSP90B1TRAP1
SCHEMBL13645718 0.78 HSP90AB1 (0.51) HSP90AB1HSP90AA1CYP2C19HSP90B1TRAP1
SCHEMBL8649570 0.77 HSP90AB1 (0.55) HSP90AB1HSP90AA1HSP90B1TRAP1HDAC6
SCHEMBL28439303 0.77 ADORA2A (0.37) HSP90AB1HSP90AA1
SCHEMBL10917478 0.77 HSP90AB1 (0.50) HSP90AB1HSP90AA1HSP90B1TRAP1HDAC6
SCHEMBL9116660 0.77 HSP90AB1 (0.46) HSP90AB1HSP90AA1HSP90B1TRAP1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6806375-B2 SUCH AS FAMCICLOVIR AND PENCICLOVIR; REACTING A 2-AMINOPURINE WITH A 1,1-BIS(OXYMETHYL)-1-VINYLMETHYL CARBONATE, ESTER OR PHOSPHATE IN THE PRESENCE OF A PALLADIUM(0) CATALYST NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2004-10-19 US disclosed
US-6555685-B1 Preparing purine derivatives, such as famiciclovir and penciclovir, by reacting, in the presence of a palladium catalyst and ligand; by-product inhibition; efficiency NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2003-04-29 US disclosed