SCHEMBL6771883

SCHEMBL6771883

Cc1ccccc1C(c1ccccc1)N(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.48
HTR2A P28223 3/20 0.47
HRH1 P35367 3/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C9 P11712 2/20 0.47
OPRM1 P35372 2/20 0.47
SLC22A2 O15244 1/20 0.47
SLC22A1 O15245 1/20 0.47
GRIN2D O15399 1/20 0.47
GRIN3B O60391 1/20 0.47
CHRM2 P08172 1/20 0.47
CHRM4 P08173 1/20 0.47
CHRM5 P08912 1/20 0.47
ADRA2A P08913 1/20 0.47
CHRM1 P11229 1/20 0.47
ADRA2B P18089 1/20 0.47
CHRM3 P20309 1/20 0.47
DRD1 P21728 1/20 0.47
SLC6A2 P23975 1/20 0.47
HRH2 P25021 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL674996 0.79 CHRNA7 (0.59) HTR2AHRH1ADRA2ASLC6A2SLC6A4
SCHEMBL29375707 0.77 ACP3 (0.49) ESR1HTR2AHRH1CYP2D6CYP2C9
Water SCHEMBL28355612 0.77 CHRNA7 (0.56) HTR2AHRH1ADRA2ASLC6A2SLC6A4
Hydrochloric Acid SCHEMBL11332719 0.77 CHRNA7 (0.56) HTR2AHRH1CYP2C9SLC6A2SLC6A4
Bromide SCHEMBL10595079 0.77 CHRNA7 (0.56) HTR2AHRH1ADRA2ASLC6A2SLC6A4
Bromide SCHEMBL11060583 0.76 MEN1 (0.40) HTR2AHRH1CYP2D6CYP2C9OPRM1
SCHEMBL8601848 0.74 ACP3 (0.48) ESR1HTR2AHRH1CYP2D6CYP2C9
SCHEMBL14509976 0.73 OPRM1 (0.43) ESR1HTR2AHRH1CYP2D6CYP2C9
SCHEMBL11708265 0.73 KMT2A (0.49) CYP2C9OPRM1MEN1KMT2AMAPT
SCHEMBL15239918 0.73 MEN1 (0.41) HTR2AHRH1CYP2C9CYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2444400-B1 SUBSTITUTED POLYCYCLIC CARBAMOYLPYRIDONE DERIVATIVE SHIONOGI & CO (JP) 2018-03-28 EP disclosed
US-20040167193-A1 Difluoromethyltriazolone compounds, use of the same and intermediates for the production thereof SUMITOMO CHEMICAL COMPANY, LIMITED 2004-08-26 US disclosed
US-6762197-B2 FUNGICIDES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-07-13 US disclosed
US-20030119670-A1 Difluoromethyltriazolone compounds, use of the same and intermediates for the production thereof SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2003-06-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040167193-A1 Difluoromethyltriazolone compounds, use of the same and intermediates for the production thereof CYP51A1, DPM1, CYP1A1 ESR1 3003/4885HTR2A 4427/4885HRH1 2616/4885
US-20030119670-A1 Difluoromethyltriazolone compounds, use of the same and intermediates for the production thereof CYP51A1, DPM1, CYP1A1 ESR1 3003/4885HTR2A 4427/4885HRH1 2616/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.