Bromide

Bromide

SCHEMBL11060583

Br.CN(C)C(c1ccccc1)c1ccccc1I

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 known ✓ P08172 1/20 0.32
ADRA2A known ✓ P08913 1/20 0.32
ADRA2B known ✓ P18089 1/20 0.32
CHRM3 known ✓ P20309 1/20 0.32
SLC6A2 known ✓ P23975 1/20 0.32
SLC6A4 known ✓ P31645 1/20 0.32
ADRA1A known ✓ P35348 1/20 0.32
SLC6A3 known ✓ Q01959 1/20 0.32
GRIN2A known ✓ Q12879 1/20 0.32
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
CYP2C9 P11712 2/20 0.40
MAPT P10636 1/20 0.40
CHRNA7 P36544 1/20 0.38
SRC P12931 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HTR2A P28223 4/20 0.36
HRH1 P35367 4/20 0.36
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL10595079 0.79 CHRNA7 (0.56) MEN1KMT2ACHRNA7KDM4EALDH1A1
SCHEMBL674996 0.76 CHRNA7 (0.59) MEN1KMT2ACHRNA7KDM4EALDH1A1
Bromide SCHEMBL11066191 0.76 CHRNA7 (0.50) MEN1KMT2ACYP2C9MAPTCHRNA7
SCHEMBL6771883 0.76 ESR1 (0.48) MEN1KMT2ACYP2C9MAPTCHRNA7
SCHEMBL11708265 0.74 KMT2A (0.49) MEN1KMT2ACYP2C9MAPTSRC
Hydrochloric Acid SCHEMBL11332719 0.74 CHRNA7 (0.56) MEN1KMT2ACYP2C9MAPTCHRNA7
Water SCHEMBL28355612 0.74 CHRNA7 (0.56) MEN1KMT2ACHRNA7KDM4EALDH1A1
SCHEMBL8318669 0.71 TYR (0.46) MEN1KMT2ACYP2C9MAPTKDM4E
SCHEMBL15239918 0.70 MEN1 (0.41) MEN1KMT2ACYP2C9MAPTCHRNA7
SCHEMBL16632702 0.70 SLC6A2 (0.41) KMT2ACYP2C9SRCALDH1A1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4446123-A QUATERNARY AMMONIUM, PHOSPHONIUM, OR ARSONIUM HALIDE HAHNEMANN UNIVERSITY (US) 1984-05-01 US claimed
US-4446123-A QUATERNARY AMMONIUM, PHOSPHONIUM, OR ARSONIUM HALIDE HAHNEMANN UNIVERSITY (US) 1984-05-01 US disclosed