SCHEMBL6772430

SCHEMBL6772430

CC(C)c1ccc(-n2nc(-c3ccccc3)c3c2C(C#N)C(C)(C)CC3=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 11/20 0.44
CDK2 P24941 11/20 0.44
LMNA P02545 4/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 1/20 0.40
SRC P12931 1/20 0.36
DHODH Q02127 1/20 0.35
ALDH1A1 P00352 3/20 0.34
MAPT P10636 3/20 0.33
KDM4E B2RXH2 2/20 0.33
HPGD P15428 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
CCNO P22674 1/20 0.33
CCNE1 P24864 1/20 0.33
CCNA1 P78396 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6770739 0.91 CCNA2 (0.45) CCNA2CDK2LMNAMEN1KMT2A
SCHEMBL6772549 0.88 CCNA2 (0.35) CCNA2CDK2LMNAMEN1KMT2A
SCHEMBL6775773 0.88 CCNA2 (0.39) CCNA2CDK2LMNAMEN1KMT2A
SCHEMBL6772794 0.87 CCNA2 (0.40) CCNA2CDK2MEN1KMT2AHTT
SCHEMBL6776854 0.86 PTGS1 (0.42) CCNA2CDK2LMNAMEN1KMT2A
SCHEMBL6771336 0.85 CCNA2 (0.37) CCNA2CDK2LMNAMEN1KMT2A
SCHEMBL6770531 0.85 MEN1 (0.40) CCNA2CDK2LMNAMEN1KMT2A
SCHEMBL6772109 0.84 CCNA2 (0.37) CCNA2CDK2LMNAMEN1KMT2A
SCHEMBL6770449 0.84 CCNA2 (0.41) CCNA2CDK2LMNAMEN1KMT2A
SCHEMBL6767158 0.84 CCNA2 (0.37) CCNA2CDK2LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed