SCHEMBL6774770

SCHEMBL6774770

Cc1nc2cc(NC(=O)c3ccccc3-c3ccc(C(F)(F)F)cc3)ccc2cc1C(=O)N[C@@H](c1ccccc1)c1ccccn1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MTTP P55157 16/20 0.48
SMO Q99835 1/20 0.45
APOB P04114 5/20 0.45
KLRK1 P26718 2/20 0.42
MICA Q29983 2/20 0.42
RAET1L Q5VY80 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7920131 0.87 MTTP (0.48) MTTPSMOAPOB
SCHEMBL6769177 0.83 MTTP (0.55) MTTPSMOAPOB
SCHEMBL6769200 0.82 MTTP (0.47) MTTPSMOAPOB
SCHEMBL6766297 0.82 MTTP (0.47) MTTPSMOAPOB
SCHEMBL6769957 0.80 TRPV1 (0.41) MTTPSMO
SCHEMBL6053015 0.79 MTTP (0.52) MTTPAPOB
SCHEMBL7679476 0.79 TRPV1 (0.43)
SCHEMBL6765645 0.77 MTTP (0.51) MTTPSMOAPOB
SCHEMBL6771609 0.76 SMO (0.47) MTTPSMOAPOB
SCHEMBL6770861 0.75 TRPV1 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6713489-B2 TREATMENT OF ATHEROSCLEROSIS, OBESITY, DIABETES, HYPERLIPIDEMIA, HYPERLIPOPROTEINEMIA, HYPERCHOLESTEROLEMIA, HYPERTRIGLYCERIDEMIA, HYPOALPHALIPOPROTEINEMIA, PANCREATITIS, MYOCARDIAL INFARCTION, STROKE, RESTENOSIS, OR SYNDROME X PFIZER INC 2004-03-30 US disclosed
US-20020132806-A1 7-[(4'-trifluoromethyl-biphenyl-2-carbonyl)amino]-quinoline-3-carboxylic acid amides, and methods of inhibiting the secretion of apolipoprotein B RUGGERI ROGER (US) 2002-09-19 US disclosed
US-6369075-B1 7[4′-trifluoromethyl-biphenyl-2-carbonyl)amino]-quinoline-3-carboxylic acid amides, and method of inhibiting the secretion of apolipoprotein B PFIZER, INC. 2002-04-09 US disclosed
EP-1099701-A1 7-[(4'-Trifluoromethyl-biphenyl-2-carbonyl)amino]-quinoline-3-carboxylic acid amides, and methods of inhibiting the secretion of apolipoprotein B Pfizer Products Inc. (US) 2001-05-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020132806-A1 7-[(4'-trifluoromethyl-biphenyl-2-carbonyl)amino]-quinoline-3-carboxylic acid amides, and methods of inhibiting the secretion of apolipoprotein B APOB, CETP, PNLIP MTTP 6/4885SMO 3658/4885APOB 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.