SCHEMBL6776573

SCHEMBL6776573

C=C(Br)C(=O)Nc1cc(C(=O)Nc2cc(C(=O)Nc3cc(C(=O)Nc4cn(C)c(C(=O)NCCC(N)=O)n4)n(C)c3)n(C)c2)n(C)c1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.49
HDAC2 Q92769 2/20 0.49
HDAC8 Q9BY41 2/20 0.49
HRAS P01112 13/20 0.48
ESR1 P03372 13/20 0.48
ESR2 Q92731 13/20 0.48
TOP1 P11387 2/20 0.48
KDM4E B2RXH2 1/20 0.48
POLB P06746 1/20 0.48
MAPT P10636 1/20 0.48
HIF1A Q16665 1/20 0.48
ERBB2 P04626 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6782496 0.95 HDAC1 (0.51) HDAC1HDAC2HDAC8HRASESR1
SCHEMBL6777138 0.95 HDAC1 (0.51) HDAC1HDAC2HDAC8HRASESR1
SCHEMBL6785507 0.91 HDAC1 (0.46) HDAC1HDAC2HDAC8HRASESR1
SCHEMBL7119707 0.90 HRAS (0.57) HDAC1HDAC2HDAC8HRASESR1
SCHEMBL7127221 0.90 HRAS (0.57) HDAC1HDAC2HDAC8HRASESR1
SCHEMBL6776283 0.90 HRAS (0.48) HDAC1HDAC2HDAC8HRASESR1
SCHEMBL7504035 0.88 HRAS (0.60) HDAC1HDAC2HDAC8HRASESR1
SCHEMBL3678651 0.88 HRAS (0.60) HDAC1HDAC2HDAC8HRASESR1
Hydrochloric Acid SCHEMBL3454587 0.87 KDM4E (0.60) HDAC1HDAC2HDAC8HRASESR1
SCHEMBL6781807 0.86 HDAC1 (0.49) HDAC1HDAC2HDAC8HRASESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6753316-B1 3-ACRYLAMIDOPYRAZOLE-5-CARBOXAMIDE DERIVATIVES PHARMACIA & UPJOHN S.P.A. (IT) 2004-06-22 US disclosed