SCHEMBL6785507

SCHEMBL6785507

C=C(Br)C(=O)Nc1cc(C(=O)Nc2cc(C(=O)Nc3cc(C(=O)Nc4cn(C)c(C(=O)NCCC(N)=NO)n4)n(C)c3)n(C)c2)n(C)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
TOP1 P11387 2/20 0.46
HRAS P01112 14/20 0.46
ESR1 P03372 13/20 0.46
ESR2 Q92731 13/20 0.46
KDM4E B2RXH2 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
HIF1A Q16665 1/20 0.45
ERBB2 P04626 1/20 0.36
EP300 Q09472 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6781807 0.96 HDAC1 (0.49) HDAC1HDAC2HDAC8TOP1HRAS
SCHEMBL6776711 0.96 HDAC1 (0.49) HDAC1HDAC2HDAC8TOP1HRAS
SCHEMBL6781649 0.91 HDAC1 (0.42) HDAC1HDAC2HDAC8TOP1HRAS
SCHEMBL6775707 0.91 HDAC1 (0.44) HDAC1HDAC2HDAC8TOP1HRAS
SCHEMBL6776573 0.91 HDAC1 (0.49) HDAC1HDAC2HDAC8TOP1HRAS
SCHEMBL7116979 0.91 HRAS (0.53) HDAC1HDAC2HDAC8TOP1HRAS
SCHEMBL7123705 0.91 HRAS (0.53) HDAC1HDAC2HDAC8TOP1HRAS
SCHEMBL6785845 0.87 HDAC1 (0.49) HDAC1HDAC2HDAC8TOP1HRAS
SCHEMBL6780417 0.87 TOP1 (0.47) HDAC1HDAC2HDAC8TOP1HRAS
Hydrochloric Acid SCHEMBL6782682 0.87 KDM4E (0.49) HDAC1HDAC2HDAC8TOP1HRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6753316-B1 3-ACRYLAMIDOPYRAZOLE-5-CARBOXAMIDE DERIVATIVES PHARMACIA & UPJOHN S.P.A. (IT) 2004-06-22 US disclosed