SCHEMBL6777843

SCHEMBL6777843

CCC(C(=O)O)C(N)c1cc(OC)c(OC)cc1Br

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.44
FYN P06241 1/20 0.44
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
ACHE P22303 1/20 0.40
GAA P10253 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6783358 0.81 ACHE (0.42) ACHETSHR
SCHEMBL6774969 0.78 TSHR (0.48) ACHETSHR
SCHEMBL9950759 0.73 LCK (0.53) LCKFYNCYP1A2CYP3A4CYP2C9
SCHEMBL6407738 0.73 CYP1A2 (0.45) LCKFYNCYP1A2CYP3A4CYP2C9
SCHEMBL7339310 0.71 CA1 (0.42) LCKFYNCYP1A2CYP3A4CYP2C9
Ethylene SCHEMBL6409433 0.71 CYP1A2 (0.43) LCKFYNCYP1A2CYP3A4CYP2C9
SCHEMBL6780474 0.70 TTR (0.43) CYP3A4CYP2C9CYP2C19GAATSHR
Oxalic Acid SCHEMBL5917366 0.69 HTR2A (0.41) LCKFYNACHE
SCHEMBL5846551 0.69 HTR2A (0.49) CYP1A2CYP3A4CYP2C9CYP2C19GAA
SCHEMBL8234075 0.69 KDM1A (0.46) LCKFYNCYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6831199-B1 In order to avoid bleeding side-effects when treating the conditions associated with integrin alpha v beta 3, it is beneficial to have compounds which are selective antagonists for alpha v beta 3 versus alpha IIb beta 3 G. D. SEARLE & CO. 2004-12-14 US disclosed