SCHEMBL6778288

SCHEMBL6778288

CCCOC(=O)COc1ccc2c(c1)c1c(n2Cc2cc(OC)cc(C(C)C)c2)CCCC1C(=O)NN

nearest known ligand 0.42

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.41
PLA2G2A P14555 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6772774 0.92 HTR6 (0.42) HTR6PLA2G2A
SCHEMBL6774224 0.79 PLA2G2A (0.39) PLA2G2A
SCHEMBL8576600 0.78 MEN1 (0.38) HTR6
SCHEMBL8576607 0.78 MEN1 (0.38)
SCHEMBL6699386 0.77 HTR6 (0.67) HTR6PLA2G2A
SCHEMBL6774375 0.75 HTR6 (0.48) HTR6PLA2G2A
SCHEMBL11824216 0.70 HTR6 (0.61) HTR6PLA2G2A
SCHEMBL11826210 0.69 HTR6 (0.64) HTR6PLA2G2A
SCHEMBL11826084 0.69 HTR6 (0.66) HTR6PLA2G2A
SCHEMBL6771051 0.68 PLA2G2A (0.44) HTR6PLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6713645-B1 INHIBITING SPLA2 MEDIATED RELEASE OF FATTY ACIDS FOR TREATMENT OF CONDITIONS SUCH AS SEPTIC SHOCK ELI LILLY AND COMPANY 2004-03-30 US disclosed
EP-0839806-B1 Substituted tricyclics LILLY CO ELI (US) 2003-07-09 EP disclosed
US-6177440-B1 THERAPY FOR SEPSIS SHOCK; PHOSPHOLIPASE INHBITOR ELI LILLY AND COMPANY 2001-01-23 US disclosed
EP-0952149-A2 Substituted carbazoles, process for their preparation and their use as sPLA2 inhibitiors ELI LILLY AND COMPANY (US) 1999-10-27 EP disclosed
WO-1998018464-A1 SUBSTITUTED TRICYCLICS ELI LILLY AND COMPANY (US) 1998-05-07 WO disclosed
EP-0839806-A1 Substituted tricyclics ELI LILLY AND COMPANY (US) 1998-05-06 EP disclosed