SCHEMBL6780431

SCHEMBL6780431

CCOC(=O)c1cc2cc(OC(C)=O)ccc2n1Cc1cccc(C(F)(F)F)c1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.51
PPARG P37231 11/20 0.51
F10 P00742 5/20 0.49
NOD2 Q9HC29 1/20 0.48
NOD1 Q9Y239 1/20 0.48
CCR2 P41597 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3578136 0.90 PPARG (0.54) PPARGF10NOD2NOD1CCR2
SCHEMBL12930106 0.87 NOD2 (0.58) PPARGF10NOD2NOD1CCR2
SCHEMBL6782501 0.85 ABCB11 (0.58) ABCB11F10NOD2NOD1CCR2
SCHEMBL1054163 0.85 NOD2 (0.55) PPARGF10NOD2NOD1CCR2
SCHEMBL3571653 0.85 NOD2 (0.67) PPARGF10NOD2NOD1
SCHEMBL925921 0.85 F10 (0.51) PPARGF10NOD2NOD1CCR2
SCHEMBL7087368 0.84 ABCB11 (0.52) ABCB11F10NOD2NOD1CCR2
SCHEMBL7083815 0.83 ABCB11 (0.61) ABCB11F10NOD2NOD1CCR2
SCHEMBL7084148 0.83 ABCB11 (0.61) ABCB11F10NOD2NOD1CCR2
SCHEMBL3979074 0.82 F10 (0.52) PPARGF10NOD2NOD1CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6737435-B1 ANTIINFLAMMATORY AGENTS; MONOCYTE CHEMOATTRACTANT PROTEIN-1 (MCP-1) DISEASES ASTRAZENECA AB (SE) 2004-05-18 US disclosed
EP-1150952-A1 INDOLE DERIVATIVES AND THEIR USE AS MCP-1 RECEPTOR ANTAGONISTS AstraZeneca AB (SE) 2001-11-07 EP disclosed
WO-2000046196-A1 INDOLE DERIVATIVES AND THEIR USE AS MCP-1 ANTAGONISTS ASTRAZENECA AB (SE) 2000-08-10 WO disclosed