SCHEMBL6786124

SCHEMBL6786124

O=c1[nH]nc(-c2cccc(NCCCCCN3CCC3)c2)c2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 7/20 0.48
ROCK1 Q13464 3/20 0.48
PARP1 P09874 3/20 0.45
HPGD P15428 1/20 0.44
NAMPT P43490 2/20 0.43
ATM Q13315 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
MAPT P10636 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HRH3 Q9Y5N1 2/20 0.41
RAD52 P43351 1/20 0.41
KMT2A Q03164 1/20 0.41
CYP2D6 P10635 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HTR7 P34969 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6787368 0.99 ROCK2 (0.47) ROCK2ROCK1PARP1HPGDNAMPT
SCHEMBL6787980 0.98 ROCK2 (0.50) ROCK2ROCK1PARP1HPGDNAMPT
SCHEMBL6783527 0.97 ROCK2 (0.49) ROCK2ROCK1PARP1HPGDNAMPT
SCHEMBL6788665 0.97 ROCK2 (0.49) ROCK2ROCK1PARP1HPGDNAMPT
Hydrochloric Acid SCHEMBL6788510 0.96 ROCK2 (0.49) ROCK2ROCK1PARP1HPGDNAMPT
Hydrochloric Acid SCHEMBL6787219 0.96 ROCK2 (0.49) ROCK2ROCK1PARP1HPGDNAMPT
SCHEMBL6782611 0.93 ROCK2 (0.46) ROCK2ROCK1PARP1HPGDNAMPT
Hydrochloric Acid SCHEMBL6786676 0.92 ROCK2 (0.45) ROCK2ROCK1PARP1HPGDNAMPT
SCHEMBL6792478 0.92 PARP1 (0.45) ROCK2ROCK1PARP1HPGDATM
SCHEMBL6783257 0.91 PARP1 (0.58) ROCK1PARP1HPGDNPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6677333-B1 ANTIISCHEMIC AGENTS; BRAIN, CARDIOVASCULAR, MUSCULAR, AND GASTROINTESTINAL DISORDERS; ANALGESICS, ANTIDIABETIC AGENTS; RETROVIRUS SENSITIZERS; ALZHEIMER*S DISEASE ONO PHARMACEUTICAL CO., LTD. (JP) 2004-01-13 US claimed
EP-1148053-A1 2H-PHTHALAZIN-1-ONE DERIVATIVES AND DRUGS COMPRISING THESE DERIVATIVES AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-10-24 EP claimed