SCHEMBL6791640

SCHEMBL6791640

O=C(NCCCn1nc2c(c1C(=O)OC(=O)C(F)(F)F)CCc1cnccc1-2)c1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
TSHR P16473 1/20 0.43
NAMPT P43490 6/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
RAB9A P51151 1/20 0.40
KMT2A Q03164 3/20 0.38
HTR1A P08908 1/20 0.38
HTR2A P28223 1/20 0.38
DRD3 P35462 1/20 0.38
USP2 O75604 1/20 0.38
MEN1 O00255 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
EPHX2 P34913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6800589 0.95 NAMPT (0.42) ALDH1A1TSHRNAMPTSMN1; SMN2HTR1A
SCHEMBL6795268 0.94 NPC1 (0.38) TSHRNAMPTSMN1; SMN2KMT2ADRD3
SCHEMBL6793648 0.88 CDK2 (0.33) RAB9AHTR2ACYP1A2CYP3A4
Trifluoroacetic Acid SCHEMBL6791633 0.88 ALDH1A1 (0.44) ALDH1A1TSHRNAMPTSMN1; SMN2RAB9A
SCHEMBL6800306 0.88 NAMPT (0.38) ALDH1A1NAMPTSMN1; SMN2KMT2AHTR1A
SCHEMBL6791548 0.87 CYP1A2 (0.33) ALDH1A1TSHRNAMPTCYP1A2CYP3A4
SCHEMBL1655698 0.87 CYP1A2 (0.30) CYP1A2CYP3A4
SCHEMBL6791910 0.87 ROCK2 (0.38) ALDH1A1TSHRNAMPTRAB9AKMT2A
SCHEMBL6794266 0.87 KMT2A (0.41) ALDH1A1TSHRSMN1; SMN2KMT2AMEN1
SCHEMBL6794582 0.86 ROCK2 (0.43) ALDH1A1SMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040127492-A1 Cyclic pyrazoles for the inhibition of mitogen activated protein kinase-activated protein kinase-2 PHARMACIA CORPORATION 2004-07-01 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040127492-A1 Cyclic pyrazoles for the inhibition of mitogen activated protein kinase-activated protein kinase-2 MKNK2, MAPKAPK2, MAP3K2 ALDH1A1 4449/4885TSHR 3404/4885NAMPT 658/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.