SCHEMBL6793264

SCHEMBL6793264

NCCC(=O)Nc1cccc(-c2n[nH]c(=O)c3ccccc23)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 6/20 0.58
ROCK2 O75116 5/20 0.58
PARP1 P09874 3/20 0.55
ATM Q13315 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
AURKA O14965 5/20 0.49
AURKB Q96GD4 4/20 0.49
MAP4K4 O95819 2/20 0.49
PIM1 P11309 2/20 0.49
RPS6KA3 P51812 2/20 0.49
STK3 Q13188 2/20 0.49
CLK4 Q9HAZ1 2/20 0.49
MAP4K5 Q9Y4K4 2/20 0.49
PRKD3 O94806 1/20 0.49
RET P07949 1/20 0.49
ROS1 P08922 1/20 0.49
PHKG2 P15735 1/20 0.49
PRKACA P17612 1/20 0.49
RPS6KB1 P23443 1/20 0.49
CDK2 P24941 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6785862 0.94 ROCK1 (0.55) ROCK1ROCK2PARP1ATMNPSR1
SCHEMBL6788685 0.93 ROCK1 (0.54) ROCK1ROCK2PARP1ATMNPSR1
SCHEMBL6782540 0.92 ROCK1 (0.53) ROCK1ROCK2PARP1ATMNPSR1
SCHEMBL6785747 0.92 ROCK1 (0.53) ROCK1ROCK2PARP1ATMNPSR1
SCHEMBL6787159 0.92 ROCK1 (0.59) ROCK1ROCK2PARP1ATMNPSR1
Hydrochloric Acid SCHEMBL6787135 0.91 ROCK1 (0.52) ROCK1ROCK2PARP1AURKAAURKB
SCHEMBL6782812 0.91 PARP1 (0.67) ROCK1ROCK2PARP1ATMNPSR1
SCHEMBL6787932 0.90 ROCK1 (0.55) ROCK1ROCK2PARP1ATMNPSR1
SCHEMBL6782196 0.88 ROCK1 (0.53) ROCK1ROCK2PARP1ATMNPSR1
SCHEMBL6786459 0.88 ROCK2 (0.53) ROCK1ROCK2PARP1ATMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6677333-B1 ANTIISCHEMIC AGENTS; BRAIN, CARDIOVASCULAR, MUSCULAR, AND GASTROINTESTINAL DISORDERS; ANALGESICS, ANTIDIABETIC AGENTS; RETROVIRUS SENSITIZERS; ALZHEIMER*S DISEASE ONO PHARMACEUTICAL CO., LTD. (JP) 2004-01-13 US claimed
EP-1148053-A1 2H-PHTHALAZIN-1-ONE DERIVATIVES AND DRUGS COMPRISING THESE DERIVATIVES AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-10-24 EP claimed
US-6677333-B1 ANTIISCHEMIC AGENTS; BRAIN, CARDIOVASCULAR, MUSCULAR, AND GASTROINTESTINAL DISORDERS; ANALGESICS, ANTIDIABETIC AGENTS; RETROVIRUS SENSITIZERS; ALZHEIMER*S DISEASE ONO PHARMACEUTICAL CO., LTD. (JP) 2004-01-13 US disclosed
EP-1148053-A1 2H-PHTHALAZIN-1-ONE DERIVATIVES AND DRUGS COMPRISING THESE DERIVATIVES AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-10-24 EP disclosed