SCHEMBL6794727

SCHEMBL6794727

NC(=O)C(NC1Cc2ccccc2C1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM7 Q14831 3/20 0.51
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
HRH3 Q9Y5N1 1/20 0.40
OPRM1 P35372 1/20 0.40
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
CCR2 P41597 1/20 0.39
ROCK2 O75116 1/20 0.39
MAPT P10636 1/20 0.39
XIAP P98170 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
PDGFRA P16234 1/20 0.38
MAPK1 P28482 1/20 0.38
MAPKAPK2 P49137 1/20 0.38
RPS6KA1 Q15418 1/20 0.38
AURKB Q96GD4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6644702 0.87 GRM7 (0.54) GRM7CA1CA2HRH3MTNR1A
SCHEMBL5097175 0.85 OPRM1 (0.48) OPRM1ROCK2MAPTMEN1KMT2A
SCHEMBL6639610 0.81 GRM7 (0.52) GRM7HRH3MTNR1AMTNR1BROCK2
SCHEMBL3315249 0.81 MEN1 (0.41) OPRM1MEN1KMT2ACYP3A4CYP2C9
SCHEMBL9282167 0.81 GAA (0.51) OPRM1MAPTMEN1KMT2ACYP3A4
SCHEMBL3313904 0.79 OPRM1 (0.42) OPRM1MEN1KMT2ACYP3A4CYP2C9
SCHEMBL7139021 0.77 KDM1A (0.53) GRM7CA1CA2HRH3MTNR1A
Hydrochloric Acid SCHEMBL6052700 0.75 KDM1A (0.51) GRM7CA1CA2HRH3MTNR1A
SCHEMBL10447052 0.73 GRM7 (0.53) GRM7CA1CA2HRH3MTNR1A
Hydrochloric Acid SCHEMBL7144136 0.73 MAPT (0.44) GRM7CA1CA2HRH3MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6743794-B2 MULTIDRUG RESISTANCE PROTEIN; CANCER; 3-(9-CHLORO-3-METHYL-4-OXO-5H-ISOXAZOLO(4,3-C)QUINOLIN-5-YL)) CYCLOHEXYL)-2-PIPERIDYLACETAMIDE ELI LILLY AND COMPANY 2004-06-01 US disclosed