SCHEMBL6796071

SCHEMBL6796071

O=C(Cc1ccccn1)NO

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.55
PDE1A P54750 1/20 0.55
PDE1B Q01064 1/20 0.55
PDE1C Q14123 1/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
POLB P06746 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA5A P35218 1/20 0.54
CA7 P43166 1/20 0.54
CA5B Q9Y2D0 1/20 0.54
HDAC6 Q9UBN7 3/20 0.52
HDAC8 Q9BY41 2/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
RAB9A P51151 2/20 0.51
NPC1 O15118 1/20 0.51
GLS O94925 4/20 0.51
HDAC1 Q13547 3/20 0.50
HDAC3 O15379 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29672808 0.83 CA1 (0.56) SMN1; SMN2POLBCA1CA2CA5A
SCHEMBL1032275 0.83 SMN1; SMN2 (0.53) SMN1; SMN2POLBCA1CA2CA5A
SCHEMBL24015947 0.83 SMN1; SMN2 (0.53) SMN1; SMN2POLBCA1CA2CA5A
SCHEMBL966286 0.83 CA1 (0.56) SMN1; SMN2POLBCA1CA2CA5A
Potassium Ion SCHEMBL11394989 0.81 CA1 (0.55) SMN1; SMN2POLBCA1CA2CA5A
Hydrochloric Acid SCHEMBL11689290 0.81 CA1 (0.55) SMN1; SMN2POLBCA1CA2CA5A
SCHEMBL2028409 0.80 CA1 (0.69) SMN1; SMN2POLBCA1CA2CA5A
SCHEMBL5032696 0.80 POLB (0.58) SMN1; SMN2POLBCA1CA2CA5A
SCHEMBL4579337 0.80 HDAC1 (0.54) SMN1; SMN2POLBHDAC6HDAC8MEN1
SCHEMBL2142240 0.79 RAB9A (0.58) SMN1; SMN2POLBCA1CA2CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0060144-A2 Cephalosporin antibiotics ELI LILLY AND COMPANY (US) 1982-09-15 EP claimed
US-6743794-B2 MULTIDRUG RESISTANCE PROTEIN; CANCER; 3-(9-CHLORO-3-METHYL-4-OXO-5H-ISOXAZOLO(4,3-C)QUINOLIN-5-YL)) CYCLOHEXYL)-2-PIPERIDYLACETAMIDE ELI LILLY AND COMPANY 2004-06-01 US disclosed
EP-0060144-A2 Cephalosporin antibiotics ELI LILLY AND COMPANY (US) 1982-09-15 EP disclosed
US-4336253-A Cephalosporin antibiotics ELI LILLY AND COMPANY (US) 1982-06-22 US disclosed