SCHEMBL6798263

SCHEMBL6798263

CCc1cc([C@H]2O[C@@H](n3cnc4c(N[C@H]5CCC[C@@H]5O)nc(Cl)nc43)[C@@H](O)[C@H]2O)on1

nearest known ligand 0.66

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.66
ADORA3 P0DMS8 10/20 0.53
ADORA1 P30542 8/20 0.53
ADORA2B P29275 6/20 0.53
MEN1 O00255 1/20 0.51
CYP1A2 P05177 1/20 0.51
MAPK1 P28482 1/20 0.51
KMT2A Q03164 1/20 0.51
RXFP1 Q9HBX9 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6576785 1.00 ADORA2A (0.66) ADORA2AADORA3ADORA1ADORA2BMEN1
SCHEMBL6573936 0.93 ADORA2A (0.69) ADORA2AADORA3ADORA1ADORA2BMEN1
SCHEMBL6572752 0.89 ADORA2A (0.51) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL6576982 0.88 ADORA2A (0.64) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL6575216 0.86 ADORA3 (0.59) ADORA2AADORA3ADORA1ADORA2BMEN1
SCHEMBL3914182 0.84 ADORA3 (0.58) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL3914192 0.84 ADORA3 (0.58) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL8090571 0.84 ADORA3 (0.58) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL6574586 0.82 ADORA3 (0.52) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL6575072 0.81 ADORA3 (0.54) ADORA2AADORA3ADORA1ADORA2BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6677316-B2 TREATING ISCHEMIA, CARDIOVASCULAR DISORDERS, STROKE, PAIN, NERVOUS SYSTEM DISORDERS OR SLEEP APNEA; ADENOSINE A1 RECEPTOR AGONIST; 2-(3-(TERT-BUTYL)-1,2,4-OXADIAZOL-5-YL)-5-(6-(ISOBUTYLAMINO)-9H-PURIN-9-YL) TETRAHYDROFURAN-3,4-DIOL SMITHKLINE BEECHAM CORPORATION 2004-01-13 US claimed