SCHEMBL6799206

SCHEMBL6799206

N#Cc1ccc(N(Cc2ccc(O)cc2)c2cnccn2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 11/20 0.49
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
HPGD P15428 1/20 0.44
CYP2C19 P33261 1/20 0.44
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
CA12 O43570 1/20 0.40
CA2 P00918 1/20 0.40
CA3 P07451 1/20 0.40
CA6 P23280 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PDK1 Q15118 1/20 0.39
MMP3 P08254 1/20 0.37
POLB P06746 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27545528 0.88 ALDH1A1 (0.44) CYP19A1KDM4EALDH1A1CYP1A2CYP2D6
SCHEMBL6802968 0.81 CYP19A1 (0.56) CYP19A1ESR1ESR2CA12CA2
SCHEMBL6799976 0.81 CYP19A1 (0.50) CYP19A1ESR1ESR2CA12CA2
SCHEMBL6797228 0.81 ESR1 (0.61) CYP19A1ESR1ESR2CA12CA2
SCHEMBL6800386 0.80 CYP19A1 (0.54) CYP19A1ESR1ESR2CA12CA2
SCHEMBL6801901 0.80 CYP19A1 (0.56) CYP19A1CA12CA2CA9
SCHEMBL6801305 0.76 CYP19A1 (0.55) CYP19A1ESR1ESR2CA12CA2
SCHEMBL6799479 0.71 CYP19A1 (0.50) CYP19A1ESR1ESR2CA12CA2
SCHEMBL8328066 0.71 CYP19A1 (0.44) CYP19A1KDM4EALDH1A1CYP1A2CYP2D6
SCHEMBL6798025 0.69 CYP19A1 (0.57) CYP19A1ESR1ESR2CA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1308297-C Phenyl sulfamate derivs. TEIKOKU HORMONE MFG CO LTD (JP) 2007-04-04 CN disclosed
US-6762205-B1 STEROID SULFATASE INHIBITORS WITHOUT ESTROGENIC SIDE EFFECT ACTION TEIKOKU HORMONE MFG. CO., LTD. (JP) 2004-07-13 US disclosed
CN-1360570-A Phenyl sulfamate derivs. TEIKOKU HORMONE MFG CO LTD (JP) 2002-07-24 CN disclosed
EP-1193250-A1 PHENYL SULFAMATE DERIVATIVES Teikoku Hormone Mfg. Co., Ltd. (JP) 2002-04-03 EP disclosed