SCHEMBL6802476

SCHEMBL6802476

O=C1CCCN1c1cccc(-n2cnc3cc(Br)cnc32)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C9 P11712 2/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
MEN1 O00255 6/20 0.40
KMT2A Q03164 6/20 0.40
GAA P10253 1/20 0.40
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
TSHR P16473 1/20 0.38
HTR6 P50406 1/20 0.38
KDM4E B2RXH2 2/20 0.37
LMNA P02545 2/20 0.37
HTT P42858 1/20 0.37
BRD4 O60885 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6803894 0.80 NT5E (0.44) HPGDCYP3A4CYP2C9ALDH1A1CYP1A2
SCHEMBL13202017 0.74 KMT2A (0.52) HPGDMEN1KMT2ASMN1; SMN2
SCHEMBL6804444 0.74 FGFR1 (0.55) HPGDMEN1KMT2A
SCHEMBL29930250 0.73 ALDH1A1 (0.62) HPGDCYP3A4CYP2C9ALDH1A1CYP1A2
SCHEMBL1634757 0.73 ALDH1A1 (0.62) HPGDCYP3A4CYP2C9ALDH1A1CYP1A2
SCHEMBL6801219 0.72 FGFR1 (0.57) HPGDALDH1A1SMN1; SMN2LMNAHTT
SCHEMBL6799091 0.71 IDO1 (0.46) HPGDCYP3A4MEN1KMT2A
SCHEMBL14910623 0.70 NPC1 (0.51) HPGDCYP3A4CYP2C9ALDH1A1CYP1A2
SCHEMBL19350803 0.69 FGFR1 (0.43) HPGDALDH1A1KMT2ASMN1; SMN2HTT
SCHEMBL29623847 0.69 FGFR1 (0.43) HPGDALDH1A1KMT2ASMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6723735-B1 TREATMENT OR PREVENTION OF ANXIETY MERCK SHARP & DOHME LTD. 2004-04-20 US disclosed
EP-1214319-B1 IMIDAZO-PYRIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME (GB) 2003-11-26 EP disclosed