SCHEMBL68043

SCHEMBL68043

Cn1cc(C(=O)Nc2ccc(F)cc2-c2ccc(Cl)c(Cl)c2)c(C(F)F)n1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 16/20 0.51
CHRM2 P08172 5/20 0.45
CHRM1 P11229 5/20 0.45
ALOX15 P16050 1/20 0.39
LMNA P02545 1/20 0.39
THRB P10828 1/20 0.39
MET P08581 1/20 0.39
AXL P30530 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29349968 1.00 CHRM3 (0.51) CHRM3CHRM2CHRM1ALOX15LMNA
SCHEMBL29445383 1.00 CHRM3 (0.51) CHRM3CHRM2CHRM1ALOX15LMNA
SCHEMBL31265248 0.93 CHRM3 (0.51) CHRM3CHRM2CHRM1
SCHEMBL1136276 0.93 CHRM3 (0.51) CHRM3CHRM2CHRM1
SCHEMBL29688317 0.93 CHRM3 (0.51) CHRM3CHRM2CHRM1ALOX15
SCHEMBL303047 0.93 CHRM3 (0.51) CHRM3CHRM2CHRM1ALOX15
SCHEMBL19274807 0.92 CHRM3 (0.45) CHRM3CHRM2CHRM1LMNATHRB
SCHEMBL1092101 0.92 CHRM3 (0.51) CHRM3CHRM2CHRM1THRB
SCHEMBL29437140 0.92 CHRM3 (0.42) CHRM3CHRM2CHRM1ALOX15LMNA
SCHEMBL304334 0.92 CHRM3 (0.42) CHRM3CHRM2CHRM1ALOX15LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1957 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4410100-A2 PLANT HEALTH COMPOSITION BASF SE (DE) 2024-08-07 EP claimed
EP-3954214-A1 MULTIPURPOSE BIOLOGICAL COMPOSITIONS Agrivalle Brasil Industria e Comércio de Produtos Agrícolas Ltda (BR) 2022-02-16 EP claimed
EP-3381289-B1 COMBINATIONS COMPRISING A FUNGICIDAL STRAIN AND AN ACTIVE COMPOUND BAYER CROPSCIENCE LP (US) 2021-05-05 EP claimed
US-10834921-B2 Foam formulations and apparatus for delivery FMC CORPORATION (US) 2020-11-17 US claimed
EP-2292098-B1 Combinations comprising a fungicidal strain and at least one additional fungicide BAYER CROPSCIENCE LP (US) 2019-11-06 EP claimed
EP-3510869-A1 COMBINATIONS COMPRISING A FUNGICIDAL STRAIN AND AN ACTIVE COMPOUND Bayer Cropscience LP (US) 2019-07-17 EP claimed
EP-2489262-B1 PESTICIDAL MIXTURES COMPRISING AN ANTHRANILAMIDE INSECTICIDE AND A FUNGICIDE BASF SE (DE) 2018-11-14 EP claimed
EP-3381289-A1 COMBINATIONS COMPRISING A FUNGICIDAL STRAIN AND AN ACTIVE COMPOUND Bayer Cropscience LP (US) 2018-10-03 EP claimed
US-20180263243-A1 NOVEL PLANT PROTECTING COMPOSITIONS AND USES THEREOF FLECHSIG PATENT COMPANY LLC (CH) 2018-09-20 US claimed
US-9844220-B2 Synergistic fungicidal active substance combinations FMC CORPORATION (US) 2017-12-19 US claimed
WO-2007031507-A1 FUNGICIDE COMPOSITION COMPRISING AN ARYLAMIDINE DERIVATIVE AND TWO KNOWN FUNGICIDE COMPOUNDS BAYER CROPSCIENCE AG (DE) 2007-03-22 WO claimed
WO-2007031141-A1 SYNERGISTIC FUNGICIDAL ACTIVE SUBSTANCE COMBINATIONS CONTAINING A CARBOXAMIDE, AN AZOLE, A SECOND AZOLE OR A STROBILURINE BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2007-03-22 WO claimed
US-20070060579-A1 Synergistic fungicidal active substance combinations BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2007-03-15 US claimed
EP-1751109-A1 FUNGICIDAL COMPOSITION COMPRISING A PYRIDYLETHYLBENZAMIDE DERIVATIVE AND A COMPOUND CAPABLE OF INHIBITING THE TRANSPORT OF ELECTRONS OF THE RESPIRATORY CHAIN IN PHYTOPATHOGENIC FUNGAL ORGANISMS Bayer CropScience S.A. (FR) 2007-02-14 EP claimed
EP-1742533-A1 USE OF ALKYKL CARBOXYLIC ACID AMIDES AS PENETRATION PROMOTERS Bayer CropScience Aktiengesellschaft (DE) 2007-01-17 EP claimed
WO-2006136551-A1 FUNGICIDE COMPOSITION COMPRISING A PHOSPHOROUS ACID DERIVATIVE, A MANDELAMIDE TYPE COMPOUND AND A FURTHER FUNGICIDE COMPOUND BAYER CROPSCIENCE SA (FR) 2006-12-28 WO claimed
WO-2006131230-A2 ACTIVE SUBSTANCE COMBINATIONS BAYER CROPSCIENCE AG (DE) 2006-12-14 WO claimed
WO-2006032356-A1 SYNERGISTIC FUNGICIDAL ACTIVE SUBSTANCE COMBINATIONS WHICH CONTAIN SPIROXAMINE, A TRIAZOLE AND A CARBOXAMIDE BAYER CROPSCIENCE AG (DE) 2006-03-30 WO claimed
WO-2005104844-A1 USE OF ALKYKL CARBOXYLIC ACID AMIDES AS PENETRATION PROMOTERS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2005-11-10 WO claimed
WO-2005077901-A1 FUNGICIDAL COMPOSITION COMPRISING A PYRIDYLETHYLBENZAMIDE DERIVATIVE AND A COMPOUND CAPABLE OF INHIBITING THE TRANSPORT OF ELECTRONS OF THE RESPIRATORY CHAIN IN PHYTOPATHOGENIC FUNGAL ORGANISMS BAYER CROPSCIENCE SA (FR) 2005-08-25 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070060579-A1 Synergistic fungicidal active substance combinations CYP51A1, CYP1A2, CYP4X1 CHRM3 94/4885CHRM2 111/4885CHRM1 122/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.