SCHEMBL6804373

SCHEMBL6804373

CCOC(=O)c1cccc2[nH]c(-c3ccc4[nH]cnc4c3)nc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.58
MAP4K4 O95819 3/20 0.53
PIM1 P11309 3/20 0.53
PIM3 Q86V86 3/20 0.53
AURKB Q96GD4 3/20 0.53
CLK4 Q9HAZ1 3/20 0.53
STK17A Q9UEE5 3/20 0.53
MAP4K5 Q9Y4K4 3/20 0.53
CLK2 P49760 2/20 0.53
MAP4K2 Q12851 2/20 0.53
DYRK1A Q13627 2/20 0.53
PRKD2 Q9BZL6 2/20 0.53
PRKD3 O94806 1/20 0.53
CAMK2D Q13557 1/20 0.53
PKN2 Q16513 3/20 0.47
PKN1 Q16512 2/20 0.47
KMT2A Q03164 1/20 0.46
ATM Q13315 1/20 0.46
PLA2G2A P14555 1/20 0.44
ALOX15 P16050 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7474098 0.84 PARP1 (0.44) PARP1MAP4K4PIM1PIM3AURKB
SCHEMBL6585180 0.84 DHODH (0.63) PARP1DHODH
SCHEMBL6810723 0.83 PARP1 (0.63) PARP1MAP4K4PIM1PIM3AURKB
SCHEMBL6810480 0.82 PARP1 (0.48) PARP1PKN2PKN1DHODH
SCHEMBL6948231 0.80 PARP1 (0.69) PARP1MAP4K4PIM1PIM3AURKB
SCHEMBL6810422 0.78 PKN1 (0.76) PARP1MAP4K4PIM1PIM3AURKB
SCHEMBL6804379 0.78 ATM (0.52) PARP1PKN2PKN1KMT2AATM
SCHEMBL6585185 0.77 HPSE (0.44) PARP1DHODH
SCHEMBL3574922 0.76 PARP1 (0.56) PARP1MAP4K4PIM1PIM3AURKB
SCHEMBL31529624 0.76 PARP1 (0.59) PARP1KMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed