SCHEMBL7474098

SCHEMBL7474098

CCOC(=O)Oc1cccc2[nH]c(-c3ccc4[nH]cnc4c3)nc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.44
HPSE Q9Y251 4/20 0.42
MGAM O43451 3/20 0.41
GAA P10253 3/20 0.41
SI P14410 3/20 0.41
MGAM2 Q2M2H8 3/20 0.41
CBFB Q13951 1/20 0.40
TP53 P04637 2/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
NPC1 O15118 1/20 0.39
HPGD P15428 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAPT P10636 1/20 0.39
PKN1 Q16512 1/20 0.38
PKN2 Q16513 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6585185 0.86 HPSE (0.44) PARP1HPSEMGAMGAASI
SCHEMBL6585182 0.85 PARP1 (0.47) PARP1HPSEPKN1PKN2
SCHEMBL6804373 0.84 PARP1 (0.58) PARP1PKN1PKN2PRKD3MAP4K4
SCHEMBL7484761 0.82 HPSE (0.43) PARP1HPSEMGAMGAASI
SCHEMBL6591471 0.79 PKN1 (0.56) PARP1HPSEMGAMGAASI
SCHEMBL7820437 0.77 MMP13 (0.51) PARP1GAAALDH1A1RAB9ASMN1; SMN2
SCHEMBL4604974 0.77 PARP1 (0.46) PARP1GAAKDM4EHPGDRAB9A
SCHEMBL7815539 0.77 PARP1 (0.57) PARP1HPSEGAATP53KDM4E
SCHEMBL6585180 0.76 DHODH (0.63) PARP1
SCHEMBL6581316 0.76 MAP4K4 (0.55) PARP1PKN2MAP4K4PIM1CLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed