SCHEMBL6804417

SCHEMBL6804417

Cc1cc(CNc2ccc(C[C]=O)cc2)c2ccccc2n1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 4/20 0.48
RAB9A P51151 2/20 0.48
SMN1; SMN2 Q16637 8/20 0.46
HTT P42858 2/20 0.46
CYP1A2 P05177 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
MAPT P10636 2/20 0.44
NPC1 O15118 1/20 0.44
GAA P10253 1/20 0.44
PKM P14618 1/20 0.43
MAPK1 P28482 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
HPGD P15428 1/20 0.42
OPRK1 P41145 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3962717 0.85 SMN1; SMN2 (0.50) ALDH1A1KDM4ERAB9ASMN1; SMN2HTT
SCHEMBL3969728 0.84 CYP1A2 (0.51) ALDH1A1KDM4ERAB9ASMN1; SMN2HTT
SCHEMBL3962723 0.82 SMN1; SMN2 (0.47) ALDH1A1KDM4ERAB9ASMN1; SMN2HTT
SCHEMBL6805411 0.82 CYP1A2 (0.49) ALDH1A1KDM4ERAB9ASMN1; SMN2HTT
SCHEMBL3970733 0.80 SMN1; SMN2 (0.47) ALDH1A1KDM4ERAB9ASMN1; SMN2HTT
SCHEMBL3970739 0.80 NCF1 (0.51) ALDH1A1KDM4ERAB9ASMN1; SMN2HTT
SCHEMBL3970289 0.78 SMN1; SMN2 (0.47) ALDH1A1KDM4ERAB9ASMN1; SMN2HTT
SCHEMBL3970211 0.78 ADAM17 (0.57)
SCHEMBL6805409 0.72 CYP1A2 (0.44) ALDH1A1KDM4ERAB9ASMN1; SMN2HTT
SCHEMBL3964963 0.72 CYP1A2 (0.50) ALDH1A1RAB9ASMN1; SMN2HTTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6770647-B2 Bicyclic hydroxamates as inhibitors of matrix metalloproteinases and/or TNF-α converting enzyme (TACE) BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-08-03 US disclosed
WO-2003016248-A2 BICYCLIC HYDROXAMATES AS INHIBITORS OF MATRIX METALLOPROTEINASES AND/OR TNF-$G(A) CONVERTING ENZYME (TACE) BRISTOL-MYERS SQUIBB COMPANY PATENT DEPARTMENT (US) 2003-02-27 WO disclosed