SCHEMBL6805072

SCHEMBL6805072

COc1ccc2[nH]cc(-c3nc4c(C(N)=O)cccc4[nH]3)c2c1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.65
PLA2G2A P14555 1/20 0.64
ALOX15 P16050 1/20 0.64
PTGS2 P35354 1/20 0.64
PKN1 Q16512 1/20 0.53
PKN2 Q16513 1/20 0.53
CHEK2 O96017 1/20 0.52
DHODH Q02127 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6585146 0.86 PARP1 (0.47) PARP1PLA2G2AALOX15PTGS2DHODH
SCHEMBL6805081 0.84 PARP1 (0.48) PARP1PLA2G2AALOX15PTGS2
SCHEMBL6807494 0.84 PARP1 (0.63) PARP1PKN1PKN2CHEK2DHODH
SCHEMBL6802028 0.83 PARP1 (0.66) PARP1PKN1PKN2CHEK2DHODH
SCHEMBL6810193 0.80 PARP1 (0.55) PARP1PLA2G2AALOX15PTGS2PKN1
SCHEMBL4321727 0.79 PARP1 (1.00) PARP1PLA2G2AALOX15PTGS2PKN1
SCHEMBL7319077 0.79 PARP1 (1.00) PARP1PLA2G2AALOX15PTGS2PKN1
SCHEMBL3117270 0.76 ATP4A (0.46) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL3633587 0.74 NR4A2 (0.73)
SCHEMBL14023455 0.73 NOX1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed