SCHEMBL6805315

SCHEMBL6805315

Cc1c(-c2nc3cccc(C(N)=O)c3[nH]2)noc1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.41
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
DHODH Q02127 2/20 0.40
BRD4 O60885 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
PTGS1 P23219 1/20 0.37
IP6K1 Q92551 1/20 0.37
S1PR1 P21453 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6805307 0.83 PARP1 (0.65) PARP1DHODH
SCHEMBL6806933 0.80 PARP1 (0.39) PARP1DHODHBRD4NPC1RAB9A
SCHEMBL3579908 0.80 PARP1 (0.61) PARP1GAADHODHNPC1RAB9A
SCHEMBL6805469 0.76 NPC1 (0.43) PARP1MEN1KMT2ADHODHBRD4
SCHEMBL29696369 0.74 NPC1 (0.53) PARP1DHODHNPC1RAB9ACYP3A4
SCHEMBL6800084 0.73 PARP1 (0.44) PARP1MEN1KMT2ADHODHRAB9A
SCHEMBL6805349 0.72 PARP1 (0.42) PARP1BRD4
SCHEMBL6805519 0.72 ALDH1A1 (0.48) PARP1DHODHNPC1RAB9A
SCHEMBL6587155 0.72 PARP1 (0.44) PARP1DHODHPTGS1
SCHEMBL6804274 0.72 PARP1 (0.69) PARP1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed