SCHEMBL6807059

SCHEMBL6807059

CC(C)(C)OC(=O)NCc1cccc(CNc2ncnc3c2ncn3CC(NC(=O)OCc2ccccc2)C(=O)OC(C)(C)C)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.45
RAB9A P51151 2/20 0.44
KMT2A Q03164 2/20 0.44
TMIGD3 P0DMS9 1/20 0.44
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44
CDK1 P06493 3/20 0.43
CCNB2 O95067 2/20 0.43
CCNB1 P14635 2/20 0.43
CCNB3 Q8WWL7 2/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
SYK P43405 1/20 0.43
ITGB3 P05106 2/20 0.42
ITGAV P06756 2/20 0.42
NPC1 O15118 1/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
AURKA O14965 1/20 0.41
RPS6KB1 P23443 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4640030 1.00 TDP1 (0.45) TDP1RAB9AKMT2ATMIGD3ADORA2A
SCHEMBL6804204 0.95 ITGB3 (0.47) TDP1RAB9AKMT2ATMIGD3ADORA2A
SCHEMBL6804197 0.95 ITGB3 (0.47) TDP1RAB9AKMT2ATMIGD3ADORA2A
SCHEMBL6016455 0.84 HDAC6 (0.43) SYKITGB3ITGAV
SCHEMBL6016459 0.84 HDAC6 (0.43) SYKITGB3ITGAV
SCHEMBL6804208 0.83 CDK1 (0.49) TDP1RAB9AKMT2ACDK1CCNB2
SCHEMBL4641283 0.83 ITGB3 (0.46) TDP1RAB9AKMT2ATMIGD3ADORA2A
SCHEMBL4640796 0.83 ITGB3 (0.47) TDP1RAB9AKMT2ATMIGD3ADORA2A
SCHEMBL4640793 0.83 ITGB3 (0.47) TDP1RAB9AKMT2ATMIGD3ADORA2A
SCHEMBL6805719 0.81 BTK (0.42) KMT2AADORA1SYKITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6723727-B1 VITRONECTIN RECEPTOR ANTAGONISTS; INHIBITORS OF BONE RESORPTION; OSTEOPOROSIS HOECHST AKTIENGESELLSCHAFT (DE) 2004-04-20 US disclosed