SCHEMBL4640796

SCHEMBL4640796

NCc1cccc(CNc2ncnc3c2ncn3C[C@@H](NC(=O)OCc2ccccc2)C(=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.47
ITGAV P06756 2/20 0.47
RAB9A P51151 2/20 0.46
KMT2A Q03164 1/20 0.46
TMIGD3 P0DMS9 1/20 0.46
ADORA2A P29274 1/20 0.46
ADORA1 P30542 1/20 0.46
NPC1 O15118 1/20 0.45
HPGD P15428 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CDK1 P06493 3/20 0.44
CCNB2 O95067 2/20 0.44
CCNB1 P14635 2/20 0.44
CCNB3 Q8WWL7 2/20 0.44
IARS1 P41252 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HUWE1 Q7Z6Z7 1/20 0.44
MARS1 P56192 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4640793 1.00 ITGB3 (0.47) ITGB3ITGAVRAB9AKMT2ATMIGD3
SCHEMBL4641283 0.90 ITGB3 (0.46) ITGB3ITGAVRAB9AKMT2ATMIGD3
SCHEMBL6804197 0.87 ITGB3 (0.47) ITGB3ITGAVRAB9AKMT2ATMIGD3
SCHEMBL6804204 0.87 ITGB3 (0.47) ITGB3ITGAVRAB9AKMT2ATMIGD3
SCHEMBL4641275 0.84 ITGB3 (0.43) ITGB3ITGAVRAB9AKMT2ATMIGD3
SCHEMBL4640030 0.83 TDP1 (0.45) ITGB3ITGAVRAB9AKMT2ATMIGD3
SCHEMBL6807059 0.83 TDP1 (0.45) ITGB3ITGAVRAB9AKMT2ATMIGD3
SCHEMBL6802305 0.82 CDK1 (0.51) CDK1CCNB2CCNB1CCNB3HUWE1
SCHEMBL5840142 0.80 HDAC6 (0.47) ITGB3ITGAV
SCHEMBL4640279 0.79 ITGB3 (0.48) ITGB3ITGAVADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853084-B1 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AG (DE) 2008-08-13 EP disclosed
US-6723727-B1 VITRONECTIN RECEPTOR ANTAGONISTS; INHIBITORS OF BONE RESORPTION; OSTEOPOROSIS HOECHST AKTIENGESELLSCHAFT (DE) 2004-04-20 US disclosed
EP-0853084-A2 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AKTIENGESELLSCHAFT (DE) 1998-07-15 EP disclosed