SCHEMBL6809503

SCHEMBL6809503

CN(CCN(C)C(=O)OC(C)(C)C)Cc1nc2ccccc2n1Cc1ccc(F)cc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.52
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
POLB P06746 2/20 0.44
TBXA2R P21731 4/20 0.44
ALOX5AP P20292 2/20 0.44
TP53 P04637 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
GNRHR P30968 1/20 0.43
CYP2D6 P10635 3/20 0.43
HRH1 P35367 3/20 0.43
KCNH2 Q12809 3/20 0.43
AGTR1 P30556 2/20 0.42
AGTR2 P50052 2/20 0.42
DRD2 P14416 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6809443 0.95 RAB9A (0.50) RAB9AHDAC1HDAC6POLBTBXA2R
SCHEMBL6813431 0.85 RAB9A (0.46) RAB9ATP53SMN1; SMN2ALDH1A1LMNA
SCHEMBL6809445 0.84 RAB9A (0.48) RAB9AHDAC1HDAC6POLBTBXA2R
SCHEMBL6809501 0.83 RAB9A (0.51) RAB9AHDAC1HDAC6POLBTBXA2R
SCHEMBL6817787 0.81 RAB9A (0.44) RAB9AHDAC1HDAC6TP53SMN1; SMN2
Hydrochloric Acid SCHEMBL6815323 0.77 RAB9A (0.45) RAB9AHDAC1HDAC6POLBTP53
SCHEMBL6817794 0.76 RAB9A (0.43) RAB9APOLBTP53SMN1; SMN2ALDH1A1
SCHEMBL6813430 0.75 RAB9A (0.45) RAB9APOLBALOX5APTP53SMN1; SMN2
SCHEMBL31504944 0.73 ACKR3 (0.53) HDAC6ALDH1A1NPSR1
Hydrochloric Acid SCHEMBL6812297 0.73 RAB9A (0.43) RAB9AHDAC1HDAC6POLBTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0980359-B1 BENZIMIDAZOLE DERIVATIVE NISSAN CHEMICAL IND LTD (JP) 2004-06-23 EP disclosed
US-6114369-A N-METHYL-N-(1-(4-FLUOROBENZYL)BENZIONIDAZOL-2-YL)-N'-METHYL-N-(3,5 -BIS(TRIFLUOROMETHYL)BENZYLAMINOCARBONYL)-1,3-PROPYLENEDIAMINE HYDROCHLORIDE, FOR EXAMPLE; SUBSTANCE P ANTAGONISTS; ANTIALLERGIC ACTIVITY NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2000-09-05 US disclosed