SCHEMBL6810012

SCHEMBL6810012

O=C(O)[C@@H]1CC(OC(=O)[C@@H]2CCCN2)CN1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.42
ALOX15 P16050 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP2D6 P10635 1/20 0.42
SLC1A3 P43003 1/20 0.42
SLC1A2 P43004 1/20 0.42
SLC1A1 P43005 1/20 0.42
NOS2 P35228 2/20 0.38
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
SLC6A1 P30531 2/20 0.37
SLC6A11 P48066 1/20 0.37
TSHR P16473 1/20 0.37
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
SLC6A13 Q9NSD5 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17187572 1.00 CYP1A2 (0.42) CYP1A2ALOX15CYP2C19CYP2D6SLC1A3
SCHEMBL4406677 0.85 NOS2 (0.31) CYP1A2ALOX15CYP2C19CYP2D6SLC1A3
SCHEMBL19345089 0.80 CYP1A2 (0.36) CYP1A2ALOX15CYP2C19CYP2D6SLC1A3
SCHEMBL7594974 0.79 CYP2D6 (0.43) CYP1A2ALOX15CYP2C19CYP2D6SLC1A3
SCHEMBL2029661 0.79 CYP2D6 (0.43) CYP1A2ALOX15CYP2C19CYP2D6SLC1A3
SCHEMBL2029987 0.79 CYP2D6 (0.43) CYP1A2ALOX15CYP2C19CYP2D6SLC1A3
SCHEMBL5198224 0.79 CYP2D6 (0.43) CYP1A2ALOX15CYP2C19CYP2D6SLC1A3
SCHEMBL2031639 0.79 CYP2D6 (0.43) CYP1A2ALOX15CYP2C19CYP2D6SLC1A3
SCHEMBL7293342 0.79 CYP2D6 (0.43) CYP1A2ALOX15CYP2C19CYP2D6SLC1A3
SCHEMBL5198220 0.79 CYP2D6 (0.43) CYP1A2ALOX15CYP2C19CYP2D6SLC1A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6833489-B1 Comprises the steps of introducing a test compound into a test chimeric, Prolyl-4-hydroxylase (P4H)-gene modified, or a wild-type nematode, wherein the test chimeric nematode has a complemented prolyl-4- hydroxylase gene mutation WISCONSIN ALUMNI RESEARCH FOUNDATION 2004-12-21 US disclosed