SCHEMBL681194

SCHEMBL681194

C=C(C(C)C)[C@H](CN(C)CC1CC1)c1ccc(Br)cc1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LSS P48449 2/20 0.40
POLB P06746 2/20 0.35
ALOX5 P09917 1/20 0.33
PYCR1 P32322 1/20 0.32
HSD11B1 P28845 3/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12193966 0.88 POLB (0.35) LSSPOLBALOX5HSD11B1CYP1A2
SCHEMBL680783 0.87 LSS (0.42) LSSPOLBALOX5MEN1KMT2A
SCHEMBL12188543 0.84 LSS (0.44) LSSPOLBALOX5MEN1KMT2A
SCHEMBL2738603 0.83 LSS (0.43) LSSPOLBALOX5MEN1KMT2A
SCHEMBL681624 0.77 PYCR1 (0.40) POLBALOX5PYCR1MEN1KMT2A
SCHEMBL681349 0.76 POLB (0.39) POLBHSD11B1KMT2ACYP1A2CYP2D6
SCHEMBL12367163 0.75 POLB (0.38) LSSPOLBALOX5CYP1A2CYP2D6
SCHEMBL681415 0.72 CHRM2 (0.43) ALOX5PYCR1CYP1A2CYP2D6
SCHEMBL16131650 0.71 CYP1A2 (0.38) LSSPOLBALOX5KMT2ACYP1A2
SCHEMBL680150 0.70 HTR2A (0.43) ALOX5KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9359340-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as Akt protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2016-06-07 US disclosed
US-8063050-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2011-11-22 US disclosed