SCHEMBL681219

SCHEMBL681219

C=C(C(C)C)[C@H](CNC(C)C)c1ccc(Cl)c(OC(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.40
MAPK1 P28482 1/20 0.38
EPHX1 P07099 1/20 0.36
SLC22A3 O75751 1/20 0.36
NOTUM Q6P988 2/20 0.34
RORC P51449 2/20 0.34
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
PGK1 P00558 1/20 0.33
RPS6KB1 P23443 1/20 0.33
EPHX2 P34913 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL681430 0.88 MAPK1 (0.42) AKT1MAPK1EPHX1SLC22A3NOTUM
SCHEMBL12188435 0.87 AKT1 (0.42) AKT1MAPK1EPHX1SLC22A3NOTUM
SCHEMBL681741 0.87 KCNN4 (0.37) SLC22A3EPHX2
SCHEMBL8226056 0.86 AKT1 (0.46) AKT1MAPK1EPHX1SLC22A3NOTUM
SCHEMBL681325 0.85 PDE2A (0.47) EPHX2
SCHEMBL681158 0.82 AKT1 (0.46) AKT1AKR1C3AKR1C2RPS6KB1
SCHEMBL681719 0.81 ALDH1A1 (0.44) MAPK1ALDH1A1
SCHEMBL681539 0.80 AKT1 (0.44) AKT1MAPK1RPS6KB1ALDH1A1
SCHEMBL681191 0.80 AKT1 (0.44) AKT1MAPK1RPS6KB1ALDH1A1
SCHEMBL681686 0.80 ALDH1A1 (0.43) EPHX1EPHX2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063050-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2011-11-22 US disclosed