SCHEMBL681741

SCHEMBL681741

C=C(C(C)C)[C@H](CNC(C)C)c1ccc(F)c(OC(F)(F)F)c1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 4/20 0.37
PDE2A O00408 5/20 0.36
SLC22A3 O75751 1/20 0.36
CACNA1H O95180 1/20 0.34
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
EPHX2 P34913 2/20 0.33
GPR139 Q6DWJ6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL681325 0.91 PDE2A (0.47) PDE2ACACNA1HEPHX2GPR139
SCHEMBL681229 0.88 CACNA1H (0.38) KCNN4PDE2ASLC22A3CACNA1HADRB2
SCHEMBL681219 0.87 AKT1 (0.40) SLC22A3EPHX2
SCHEMBL12188490 0.87 KCNN4 (0.38) KCNN4PDE2ASLC22A3CACNA1HADRB2
SCHEMBL17803800 0.86 SLC22A3 (0.47) SLC22A3CACNA1HADRB2ADRB1ADRB3
SCHEMBL2739078 0.86 KCNN4 (0.39) KCNN4PDE2ASLC22A3CACNA1HADRB2
SCHEMBL680064 0.82 PDPK1 (0.44) ADRB2ADRB1ADRB3
SCHEMBL681710 0.81 AKT1 (0.45) ADRB2ADRB1ADRB3
SCHEMBL681686 0.81 ALDH1A1 (0.43) PDE2AADRB2ADRB1ADRB3EPHX2
SCHEMBL17803797 0.80 ADRB2 (0.38) ADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063050-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2011-11-22 US disclosed