SCHEMBL6812958

SCHEMBL6812958

CCOC(=O)COc1ccc(C(=O)CBr)cc1CC

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
MAPK1 P28482 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ESR1 P03372 1/20 0.43
SRD5A2 P31213 1/20 0.43
ABCB1 P08183 1/20 0.41
CASP3 P42574 1/20 0.41
CASP7 P55210 1/20 0.41
CASP9 P55211 1/20 0.41
GSK3B P49841 1/20 0.41
USP2 O75604 1/20 0.41
HPGD P15428 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
NTSR1 P30989 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2009931 0.89 ALDH1A1 (0.50) ALDH1A1L3MBTL1ESR1ABCB1CASP3
Bromide SCHEMBL5787146 0.88 ALDH1A1 (0.49) ALDH1A1L3MBTL1ESR1ABCB1CASP3
SCHEMBL7328604 0.88 ESR1 (0.52) ALDH1A1L3MBTL1ESR1ABCB1CASP3
SCHEMBL6812575 0.86 NPSR1 (0.49) ALDH1A1MAPK1L3MBTL1NPSR1LMNA
SCHEMBL6809954 0.86 GAA (0.50) ALDH1A1L3MBTL1ESR1ABCB1CASP3
SCHEMBL6813482 0.86 L3MBTL1 (0.52) ALDH1A1L3MBTL1ESR1ABCB1CASP3
SCHEMBL2012596 0.85 ALDH1A1 (0.51) ALDH1A1MAPK1L3MBTL1HPGDNPSR1
SCHEMBL7462216 0.85 ALDH1A1 (0.60) ALDH1A1MAPK1L3MBTL1SMN1; SMN2HPGD
SCHEMBL2009817 0.82 ESR1 (0.42) ALDH1A1L3MBTL1ESR1ABCB1CASP3
SCHEMBL2009646 0.81 NPC1 (0.51) ALDH1A1MAPK1L3MBTL1SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095932-B1 PHENOXYACETIC ACID DERIVATIVES AND MEDICINAL COMPOSITIONS CONTAINING THE SAME KISSEI PHARMACEUTICAL (JP) 2004-05-19 EP disclosed
US-6538152-B1 Obesity, hyperglycemia, urinary incontinence, intestinal or biliary calculi hypermotility, pollakiuria and depression treatment KISSEI PHARMACEUTICAL CO., LTD. (JP) 2003-03-25 US disclosed
EP-1095932-A1 PHENOXYACETIC ACID DERIVATIVES AND MEDICINAL COMPOSITIONS CONTAINING THE SAME Kissei Pharmaceutical Co., Ltd. (JP) 2001-05-02 EP disclosed