SCHEMBL6813645

SCHEMBL6813645

Cc1c(=O)c(Cc2ccc(F)c(F)c2)cn2nc(C(=O)O)[nH]c12.NC(=O)c1ccncc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 1/20 0.36
KDM5A P29375 2/20 0.36
KDM5B Q9UGL1 2/20 0.36
P2RY14 Q15391 1/20 0.33
VNN1 O95497 1/20 0.32
CYP17A1 P05093 1/20 0.32
KDM4C Q9H3R0 2/20 0.32
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 1/20 0.31
NCOA1 Q15788 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
PARP1 P09874 1/20 0.31
LDHA P00338 1/20 0.30
LDHB P07195 1/20 0.30
PDE2A O00408 1/20 0.30
MPO P05164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6813649 0.90 KDM5A (0.36) KDM5AKDM5BP2RY14CYP17A1KDM4E
SCHEMBL6476575 0.90 KDM5A (0.40) KDM5AKDM5BP2RY14KDM4CALDH1A1
SCHEMBL6813648 0.82 NAMPT (0.39) ALDH1A1PDE2A
SCHEMBL6478088 0.77 PTGER4 (0.41) KDM4EALDH1A1
Niacinamide SCHEMBL6818598 0.72 FYN (0.39) FYNP2RY14VNN1KDM4EMEN1
SCHEMBL6489375 0.71 GRM4 (0.33) KDM5AKDM5BMPO
SCHEMBL6485426 0.71 P2RY14 (0.36) FYNKDM5AKDM5BP2RY14PARP1
SCHEMBL6289368 0.71 KDM5A (0.38) KDM5AKDM5BP2RY14LDHALDHB
SCHEMBL6490897 0.70 KDM5A (0.38) FYNKDM5AKDM5BP2RY14MEN1
SCHEMBL6819189 0.66 KDM5A (0.37) FYNKDM5AKDM5BP2RY14KDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014908-A1 HETEROBICYLCIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO claimed