SCHEMBL6813655

SCHEMBL6813655

CCOC(=O)COc1ccc(CCBr)cc1C#N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.44
ADRB2 P07550 2/20 0.44
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
CASR P41180 2/20 0.44
SLC6A3 Q01959 2/20 0.44
KCNH2 Q12809 2/20 0.44
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
HSD17B10 Q99714 2/20 0.42
TP53 P04637 1/20 0.42
ALDH1A1 P00352 3/20 0.42
NLRP3 Q96P20 1/20 0.42
S1PR1 P21453 2/20 0.41
ABCB1 P08183 1/20 0.41
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
ADRB3 P13945 2/20 0.40
HPGD P15428 2/20 0.40
SQOR Q9Y6N5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6813895 0.89 CYP4F2 (0.49) CYP2D6ADRB2SLC6A2SLC6A4CASR
SCHEMBL6818076 0.84 CYP2D6 (0.42) CYP2D6ADRB2SLC6A2SLC6A4CASR
SCHEMBL6813642 0.83 ESR1 (0.52) HSD17B10ALDH1A1ABCB1PPARGPPARA
SCHEMBL6813693 0.82 ALDH1A1 (0.48) ALDH1A1ABCB1PPARGPPARA
SCHEMBL6813752 0.82 ALDH1A1 (0.45) HSD17B10ALDH1A1ABCB1PPARGPPARA
SCHEMBL15074081 0.82 POLB (0.48) NPC1RAB9AHSD17B10TP53ALDH1A1
SCHEMBL6813613 0.82 GAA (0.50) CYP2D6NPC1RAB9AHSD17B10ALDH1A1
SCHEMBL6813807 0.82 ESR1 (0.48) HSD17B10ALDH1A1ABCB1PPARGPPARA
SCHEMBL14026553 0.82 NPC1 (0.50) NPC1RAB9AHSD17B10TP53ALDH1A1
SCHEMBL6818105 0.81 ADRB3 (0.57) HSD17B10ALDH1A1ABCB1PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095932-B1 PHENOXYACETIC ACID DERIVATIVES AND MEDICINAL COMPOSITIONS CONTAINING THE SAME KISSEI PHARMACEUTICAL (JP) 2004-05-19 EP disclosed
US-6538152-B1 Obesity, hyperglycemia, urinary incontinence, intestinal or biliary calculi hypermotility, pollakiuria and depression treatment KISSEI PHARMACEUTICAL CO., LTD. (JP) 2003-03-25 US disclosed
EP-1095932-A1 PHENOXYACETIC ACID DERIVATIVES AND MEDICINAL COMPOSITIONS CONTAINING THE SAME Kissei Pharmaceutical Co., Ltd. (JP) 2001-05-02 EP disclosed