SCHEMBL6814

SCHEMBL6814

Cc1noc(-c2ccc(Br)cc2)c1C(CO)SCC(F)(F)F

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11802 0.82 CYP1A2 (0.33) CYP1A2CYP3A4CYP2C9CYP2C19TDP1
SCHEMBL6943 0.81 EPHX1 (0.35) CYP2C9
SCHEMBL2087 0.81 EPHX1 (0.35) CYP2C9
SCHEMBL7689 0.81 CYP1A2 (0.31) CYP1A2CYP3A4CYP2C9CYP2C19TDP1
SCHEMBL1307 0.80 EPHX1 (0.41)
SCHEMBL1627 0.80 EPHX1 (0.41)
SCHEMBL6813 0.79 TRPV1 (0.30) TRPV1
SCHEMBL7387 0.78 NR1I2 (0.35) CYP1A2CYP3A4CYP2C9CYP2C19TDP1
SCHEMBL7688 0.72 ALDH1A1 (0.35) CYP1A2CYP2C9TRPV1
SCHEMBL18597743 0.71 ALDH1A1 (0.38) CYP1A2CYP3A4CYP2C9CYP2C19TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483252-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041694-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed