SCHEMBL6816409

SCHEMBL6816409

COc1ccc(CCOc2cccc(C(=O)Nc3c(Br)cccc3C(=O)O)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 1/20 0.52
AKR1C2 P52895 2/20 0.52
AKR1C1 Q04828 2/20 0.52
NR1H4 Q96RI1 5/20 0.48
TSHR P16473 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
PKM P14618 1/20 0.45
HTT P42858 1/20 0.45
SLC2A1 P11166 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
KMT2A Q03164 1/20 0.44
PYGM P11217 1/20 0.43
MAPT P10636 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
CSNK2A2 P19784 1/20 0.43
CSNK2A1 P68400 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6349430 0.83 AKR1C2 (0.75) SMPD1AKR1C2AKR1C1NR1H4TSHR
SCHEMBL6817692 0.76 NR4A2 (0.63) SMPD1AKR1C2AKR1C1NR1H4NPC1
SCHEMBL6817166 0.75 MAOB (0.59) SMPD1AKR1C2AKR1C1NR1H4HTT
SCHEMBL202923 0.74 PARP1 (0.63) SMPD1SLC2A1ALDH1A1KMT2AMAPT
SCHEMBL6349641 0.73 PLK1 (0.60) AKR1C2AKR1C1NPSR1PKMMEN1
SCHEMBL15820015 0.70 TP53 (0.67) SMPD1NR1H4NPC1RAB9ASMN1; SMN2
SCHEMBL3630514 0.70 NR1H4 (0.59) SMPD1NR1H4HTTNPC1RAB9A
SCHEMBL7104144 0.70 NPC1 (0.53) TSHRNPC1RAB9ASMN1; SMN2MEN1
SCHEMBL15826402 0.70 KMT2A (0.60) NR1H4PKMHTTNPC1RAB9A
SCHEMBL6816406 0.69 SMPD1 (0.45) SMPD1NR1H4PKMHTTSLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004018414-A2 ANTIBACTERIAL AGENTS PHARMACIA & UPJOHN COMPANY LLC (US) 2004-03-04 WO claimed