SCHEMBL6817692

SCHEMBL6817692

O=C(Nc1c(Br)cccc1C(=O)O)c1cccc(OCc2cccc(F)c2)c1

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 3/20 0.63
MAOB P27338 3/20 0.56
SMPD1 P17405 2/20 0.52
NR1H4 Q96RI1 2/20 0.52
MRGPRX4 Q96LA9 2/20 0.51
HPD P32754 1/20 0.48
AKR1C2 P52895 1/20 0.48
AKR1C1 Q04828 1/20 0.48
NPC1 O15118 1/20 0.48
ALDH1A1 P00352 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
MAOA P21397 1/20 0.48
SIRT2 Q8IXJ6 1/20 0.48
SIRT1 Q96EB6 1/20 0.48
SIRT3 Q9NTG7 1/20 0.48
PPARA Q07869 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6812774 0.91 NR4A2 (0.62) NR4A2MAOBNR1H4MRGPRX4NPC1
SCHEMBL6817166 0.84 MAOB (0.59) MAOBSMPD1NR1H4AKR1C2AKR1C1
SCHEMBL6352870 0.84 AKR1C2 (0.70) NR4A2MAOBSMPD1NR1H4MRGPRX4
SCHEMBL27921579 0.79 NR4A2 (0.75) NR4A2MAOBSMPD1MRGPRX4HPD
SCHEMBL6816409 0.76 SMPD1 (0.52) SMPD1NR1H4AKR1C2AKR1C1NPC1
SCHEMBL6812445 0.75 MAOB (0.58) MAOBNR1H4ALDH1A1RAB9AMAOA
SCHEMBL4208795 0.74 NR4A2 (0.62) NR4A2MAOBNR1H4MRGPRX4AKR1C2
SCHEMBL15825643 0.74 SMPD1 (0.61) NR4A2MAOBSMPD1NR1H4MRGPRX4
SCHEMBL6352019 0.73 AKR1C2 (0.78) NR4A2SMPD1NR1H4MRGPRX4AKR1C2
SCHEMBL6306323 0.72 NR4A2 (0.70) NR4A2MAOBMAOAPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004018414-A2 ANTIBACTERIAL AGENTS PHARMACIA & UPJOHN COMPANY LLC (US) 2004-03-04 WO claimed