SCHEMBL6816697

SCHEMBL6816697

COc1ccccc1CC1(C#N)CCNCC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 5/20 0.51
USP2 O75604 1/20 0.51
SIGMAR1 Q99720 3/20 0.46
SLC6A2 P23975 5/20 0.44
SLC6A4 P31645 5/20 0.44
KCNH2 Q12809 4/20 0.44
SLC6A3 Q01959 3/20 0.44
HTR7 P34969 1/20 0.44
GNAI3 P08754 1/20 0.42
DRD2 P14416 2/20 0.42
HTR2C P28335 2/20 0.40
IDO1 P14902 2/20 0.38
TAAR1 Q96RJ0 1/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
ADRB1 P08588 1/20 0.38
CYP2C19 P33261 1/20 0.38
DRD3 P35462 1/20 0.38
HTR3A P46098 1/20 0.38
HTR6 P50406 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29363767 0.90 KCNH2 (0.44) CYP2D6USP2SIGMAR1KCNH2IDO1
SCHEMBL31118222 0.87 KCNH2 (0.42) CYP2D6USP2SIGMAR1KCNH2IDO1
SCHEMBL22719337 0.81 LMNA (0.43) CYP2D6USP2SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL7844991 0.79 LMNA (0.45) CYP2D6USP2SLC6A2SLC6A4SLC6A3
SCHEMBL20070372 0.78 SIGMAR1 (0.56) CYP2D6USP2SIGMAR1SLC6A2SLC6A4
SCHEMBL22728358 0.78 BACE1 (0.43) CYP2D6USP2SLC6A2SLC6A4IDO1
SCHEMBL6027203 0.78 BACE1 (0.37) CYP2D6USP2SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL28123155 0.77 SLC6A2 (0.42) CYP2D6SLC6A2SLC6A4KCNH2SLC6A3
Hydrochloric Acid SCHEMBL20138396 0.77 SIGMAR1 (0.55) CYP2D6USP2SIGMAR1SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL28123265 0.77 BACE1 (0.42) CYP2D6USP2SIGMAR1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004010942-A2 SUBSTITUTED HETEROCYCLIC COMPOUNDS AS MODULATORS OF THE CCR5 RECEPTOR SMITHKLINE BEECHAM CORPORATION (US) 2004-02-05 WO disclosed