SCHEMBL681752

SCHEMBL681752

C=C(C(C)C)[C@H](CNC(C)C)c1ccc(Cl)cc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 7/20 0.40
ADRB1 P08588 7/20 0.40
ADRB3 P13945 6/20 0.40
MDM2 Q00987 1/20 0.36
KDM4E B2RXH2 2/20 0.34
KCNH2 Q12809 1/20 0.33
LMNA P02545 1/20 0.33
S1PR3 Q99500 2/20 0.33
PYGL P06737 1/20 0.33
S1PR1 P21453 1/20 0.33
OPRM1 P35372 1/20 0.33
RAB9A P51151 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL681744 1.00 ADRB2 (0.40) ADRB2ADRB1ADRB3MDM2KDM4E
SCHEMBL679667 0.86 ADRB2 (0.40) ADRB2ADRB1ADRB3MDM2KDM4E
SCHEMBL681005 0.86 ADRB2 (0.40) ADRB2ADRB1ADRB3MDM2KDM4E
SCHEMBL681279 0.86 LMNA (0.42) ADRB2ADRB1LMNARAB9AMEN1
SCHEMBL12188385 0.85 ADRB2 (0.41) ADRB2ADRB1ADRB3MDM2KDM4E
SCHEMBL12188387 0.85 ADRB2 (0.41) ADRB2ADRB1ADRB3MDM2KDM4E
SCHEMBL17803802 0.85 ADRB2 (0.41) ADRB2ADRB1ADRB3KDM4EALDH1A1
SCHEMBL2738447 0.84 ADRB2 (0.40) ADRB2ADRB1ADRB3MDM2KDM4E
SCHEMBL8220416 0.84 ADRB2 (0.40) ADRB2ADRB1ADRB3MDM2KDM4E
SCHEMBL2738452 0.84 ADRB2 (0.40) ADRB2ADRB1ADRB3MDM2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9359340-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as Akt protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2016-06-07 US disclosed
US-8063050-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2011-11-22 US disclosed