SCHEMBL6817664

SCHEMBL6817664

COc1cc(Cl)c(-c2ccnc(NCCCC3CC3)c2N)cc1C

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT5A Q9NQR1 1/20 0.34
BRD4 O60885 2/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
CRHR1 P34998 2/20 0.33
STK17B O94768 1/20 0.33
STK17A Q9UEE5 1/20 0.33
LRRK2 Q5S007 1/20 0.33
TNF P01375 1/20 0.32
EHMT2 Q96KQ7 1/20 0.32
ACP1 P24666 1/20 0.32
ACHE P22303 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6817843 0.89 SCN9A (0.37) KMT5ACRHR1STK17BSTK17ALRRK2
SCHEMBL6817679 0.88 STK17B (0.35) KMT5ABRD4STK17BSTK17ALRRK2
SCHEMBL6817533 0.85 HSP90AA1 (0.37) KMT5AHSP90AA1HSP90AB1CRHR1ACP1
SCHEMBL6821721 0.84 NPC1 (0.34) KMT5ABRD4LRRK2ACP1
SCHEMBL6822467 0.82 KMT5A (0.34) KMT5ABRD4TNFEHMT2ACP1
SCHEMBL6818015 0.81 ACP1 (0.36) KMT5ABRD4HSP90AA1HSP90AB1CRHR1
SCHEMBL6817777 0.79 BRD4 (0.37) BRD4CRHR1
SCHEMBL6814612 0.78 BCHE (0.30) ACHE
SCHEMBL6813647 0.77 ACP1 (0.43) CRHR1ACP1
SCHEMBL6082536 0.77 IDO1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004031189-A1 PYRIDINO AND PYRIMIDINO PYRAZINONES FOR TREATMENT OF ANXIETY AND DEPRESSION BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2004-04-15 WO disclosed