SCHEMBL6817843

SCHEMBL6817843

COc1cc(Cl)c(-c2ccnc(NCCCC3CC3)c2N)cc1F

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.37
JAK1 P23458 1/20 0.35
JAK3 P52333 1/20 0.35
STK17A Q9UEE5 2/20 0.34
STK17B O94768 1/20 0.34
KMT5A Q9NQR1 1/20 0.33
BCL6 P41182 2/20 0.33
CCNT1 O60563 1/20 0.32
CDK9 P50750 1/20 0.32
LRRK2 Q5S007 1/20 0.32
TNF P01375 1/20 0.32
CRHR1 P34998 1/20 0.32
EHMT2 Q96KQ7 1/20 0.32
ACP1 P24666 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6822467 0.89 KMT5A (0.34) SCN9AKMT5ACCNT1CDK9TNF
SCHEMBL6817664 0.89 KMT5A (0.34) STK17ASTK17BKMT5ALRRK2TNF
SCHEMBL6814612 0.85 BCHE (0.30)
SCHEMBL6813930 0.84 SCN9A (0.37) SCN9AJAK1JAK3CCNT1CDK9
SCHEMBL6817533 0.84 HSP90AA1 (0.37) KMT5ACCNT1CDK9CRHR1ACP1
SCHEMBL6817679 0.83 STK17B (0.35) STK17ASTK17BKMT5ALRRK2TNF
SCHEMBL6818015 0.80 ACP1 (0.36) KMT5ACCNT1CDK9CRHR1ACP1
SCHEMBL6818651 0.78 BRD4 (0.34) SCN9AJAK1JAK3
SCHEMBL6813647 0.78 ACP1 (0.43) SCN9ACRHR1ACP1
SCHEMBL6817674 0.77 CRHR1 (0.36) CCNT1CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004031189-A1 PYRIDINO AND PYRIMIDINO PYRAZINONES FOR TREATMENT OF ANXIETY AND DEPRESSION BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2004-04-15 WO disclosed