SCHEMBL6813647

SCHEMBL6813647

Nc1c(-c2ccc(C(F)(F)F)cc2Cl)ccnc1NCCCC1CC1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 2/20 0.43
CRHR1 P34998 9/20 0.39
CRHR2 Q13324 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
NPC1 O15118 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C19 P33261 1/20 0.35
CASP3 P42574 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
SCN9A Q15858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6817533 0.83 HSP90AA1 (0.37) ACP1CRHR1CRHR2CYP1A2CYP3A4
SCHEMBL6817674 0.82 CRHR1 (0.36) CRHR1CRHR2
SCHEMBL6818015 0.80 ACP1 (0.36) ACP1CRHR1CRHR2NPC1RAB9A
SCHEMBL6818255 0.79 CRHR1 (0.36) CRHR1CRHR2
SCHEMBL6817843 0.78 SCN9A (0.37) ACP1CRHR1SCN9A
SCHEMBL6814612 0.78 BCHE (0.30)
SCHEMBL6817664 0.77 KMT5A (0.34) ACP1CRHR1
SCHEMBL6082284 0.76 NR1I2 (0.38)
SCHEMBL6817679 0.75 STK17B (0.35) SMN1; SMN2
SCHEMBL6818651 0.71 BRD4 (0.34) CYP3A4SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004031189-A1 PYRIDINO AND PYRIMIDINO PYRAZINONES FOR TREATMENT OF ANXIETY AND DEPRESSION BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2004-04-15 WO disclosed