SCHEMBL6818210

SCHEMBL6818210

Cc1cccc2c1CC(CN)(CC(=O)O)C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.39
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
TSHR P16473 1/20 0.39
BLM P54132 1/20 0.39
CACNA2D1 P54289 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KMT2A Q03164 3/20 0.36
CD69 Q07108 1/20 0.33
CXCR5 P32302 7/20 0.33
CYP2D6 P10635 3/20 0.33
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
CYP3A4 P08684 1/20 0.33
HTR1A P08908 1/20 0.33
HTR1B P28222 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR7 P34969 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7614604 0.87 KMT2A (0.36) LMNAALDH1A1TSHRBLMKMT2A
SCHEMBL6818043 0.85 ALDH1A1 (0.39) LMNAUSP2ALDH1A1CYP1A2TSHR
SCHEMBL6818099 0.85 ALDH1A1 (0.46) LMNAUSP2ALDH1A1CYP1A2TSHR
SCHEMBL14459076 0.84 ALDH1A1 (0.40) LMNAUSP2ALDH1A1CYP1A2TSHR
SCHEMBL6813335 0.84 HTR1A (0.48) LMNAUSP2ALDH1A1CYP1A2TSHR
SCHEMBL6818094 0.84 USP2 (0.40) LMNAUSP2ALDH1A1CYP1A2TSHR
SCHEMBL6817221 0.83 ALDH1A1 (0.39) LMNAUSP2ALDH1A1CYP1A2TSHR
SCHEMBL6817613 0.83 USP2 (0.39) LMNAUSP2ALDH1A1CYP1A2TSHR
SCHEMBL6813555 0.83 USP2 (0.39) LMNAUSP2ALDH1A1CYP1A2TSHR
SCHEMBL6813724 0.83 AKR1B1 (0.44) LMNAUSP2ALDH1A1CYP1A2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1180094-B1 FUSED POLYCYCLIC AMINO ACIDS AS PHARMACEUTICAL AGENTS WARNER LAMBERT CO (US) 2004-07-28 EP claimed
WO-2007090661-A2 ACTIVE SUBSTANCE COMBINATION COMPRISING AZOLYLCARBINOL COMPOUNDS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-08-16 WO disclosed
EP-1180094-B1 FUSED POLYCYCLIC AMINO ACIDS AS PHARMACEUTICAL AGENTS WARNER LAMBERT CO (US) 2004-07-28 EP disclosed