SCHEMBL6818672

SCHEMBL6818672

COc1ccc(-c2ncnc3c2nc(C)c(=O)n3CCC2CCC2)c(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 1/20 0.40
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
PIK3CA P42336 2/20 0.38
PDE2A O00408 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6822135 0.96 CRHR1 (0.42) CRHR1PIK3CA
SCHEMBL6818621 0.87 PIK3CA (0.37) CRHR1PIK3CA
SCHEMBL6817739 0.83 CYP1A2 (0.43)
SCHEMBL6814074 0.83 ERBB2 (0.47) CRHR1
SCHEMBL6821866 0.82 CRHR1 (0.39) CRHR1PIK3CA
SCHEMBL6819175 0.82 CRHR1 (0.36) CRHR1
SCHEMBL6818951 0.82
SCHEMBL6818754 0.80 CRHR1 (0.38) CRHR1
SCHEMBL6082194 0.80
SCHEMBL6082186 0.80

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004031189-A1 PYRIDINO AND PYRIMIDINO PYRAZINONES FOR TREATMENT OF ANXIETY AND DEPRESSION BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2004-04-15 WO claimed
WO-2004031189-A1 PYRIDINO AND PYRIMIDINO PYRAZINONES FOR TREATMENT OF ANXIETY AND DEPRESSION BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2004-04-15 WO disclosed