SCHEMBL6821486

SCHEMBL6821486

COCCCCn1c(=O)c(C)nc2c(Cl)ccnc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 12/20 0.46
ALDH1A1 P00352 10/20 0.46
CYP3A4 P08684 7/20 0.46
HSD17B10 Q99714 7/20 0.46
CYP2C19 P33261 4/20 0.46
CYP2C9 P11712 4/20 0.46
USP2 O75604 3/20 0.46
MAPK1 P28482 2/20 0.46
CASP1 P29466 3/20 0.44
CASP7 P55210 3/20 0.44
TSHR P16473 7/20 0.43
CLK4 Q9HAZ1 2/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
STK4 Q13043 1/20 0.40
STK3 Q13188 1/20 0.40
SIK2 Q9H0K1 1/20 0.40
STK26 Q9P289 1/20 0.40
STK24 Q9Y6E0 1/20 0.40
PDE2A O00408 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6814314 0.84
SCHEMBL6819066 0.83
SCHEMBL6814766 0.83 CYP1A2 (0.44) CYP1A2CYP3A4CYP2C19CYP2C9TSHR
SCHEMBL6818786 0.80 STK4 (0.42) STK4STK3SIK2STK26STK24
SCHEMBL6817702 0.79
SCHEMBL6814620 0.79 ALDH1A1 (0.40) CYP1A2ALDH1A1HSD17B10CASP1CASP7
SCHEMBL6818381 0.78 CYP1A2 (0.46) CYP1A2ALDH1A1CYP3A4CYP2C19CYP2C9
SCHEMBL6817739 0.76 CYP1A2 (0.43) CYP1A2ALDH1A1CYP3A4HSD17B10CYP2C19
SCHEMBL6818661 0.76 ALDH1A1 (0.39) CYP1A2ALDH1A1CYP3A4
SCHEMBL6082587 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004031189-A1 PYRIDINO AND PYRIMIDINO PYRAZINONES FOR TREATMENT OF ANXIETY AND DEPRESSION BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2004-04-15 WO disclosed