SCHEMBL6821650

SCHEMBL6821650

CC(=O)Nc1ccc(-c2cc3noc(C(=O)Nc4ccc(Br)cc4C(=O)O)c3cc2NC(C)=O)c(C(F)(F)F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK2 O95069 2/20 0.38
KCNK10 P57789 2/20 0.38
ALDH1A1 P00352 2/20 0.37
MAP2K1 Q02750 1/20 0.36
MPO P05164 2/20 0.35
PTGFR P43088 1/20 0.35
AKR1C2 P52895 4/20 0.35
AKR1C1 Q04828 3/20 0.35
AKR1C3 P42330 2/20 0.35
AKR1C4 P17516 1/20 0.35
KDM4E B2RXH2 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HTT P42858 1/20 0.34
GRIK1 P39086 1/20 0.34
S1PR1 P21453 2/20 0.34
S1PR3 Q99500 2/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
DNMT3A Q9Y6K1 1/20 0.33
SORT1 Q99523 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6833746 0.89 KCNK2 (0.39) KCNK2KCNK10ALDH1A1MAP2K1MPO
SCHEMBL6818135 0.88 RORC (0.34) MAP2K1MPOKDM4EHSD17B10S1PR1
SCHEMBL6833974 0.78 TAS2R14 (0.42) MAP2K1MPOHTTGRIK1S1PR1
SCHEMBL6833954 0.78 RORC (0.35) MAP2K1MPOKDM4EHSD17B10S1PR1
SCHEMBL6710154 0.74 GRIK1 (0.40) ALDH1A1MAP2K1HTTGRIK1S1PR1
SCHEMBL6818553 0.74 AKR1C2 (0.50) KCNK2KCNK10PTGFRAKR1C2AKR1C1
SCHEMBL6818600 0.73 TP53 (0.34) MAP2K1MPOS1PR1S1PR3
SCHEMBL6821982 0.71 TP53 (0.34) S1PR1S1PR3
SCHEMBL6818246 0.71 TP53 (0.34) MAP2K1S1PR1S1PR3
SCHEMBL6822026 0.71 EGLN2 (0.35) MAP2K1MPOS1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004018428-A1 ANTIBACTERIAL BENZOIC ACID DERIVATIVES PHARMACIA & UPJOHN COMPANY LLC (US) 2004-03-04 WO disclosed