SCHEMBL6821984

SCHEMBL6821984

CNC(=O)CCc1ccc(N(CC(=O)OC)S(=O)(=O)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 5/20 0.40
PTPN6 P29350 1/20 0.40
PTPN11 Q06124 1/20 0.40
NR1H2 P55055 1/20 0.39
CA1 P00915 5/20 0.38
CA2 P00918 4/20 0.38
CA12 O43570 3/20 0.38
CA14 Q9ULX7 3/20 0.38
ALDH1A1 P00352 3/20 0.38
CA7 P43166 2/20 0.38
NR1I2 O75469 1/20 0.35
RAB9A P51151 1/20 0.35
MLYCD O95822 1/20 0.35
MAPK1 P28482 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GLA P06280 1/20 0.34
KMT2A Q03164 1/20 0.34
POLB P06746 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6820995 0.84 SMN1; SMN2 (0.44) PTPN1PTPN6PTPN11CA1CA2
SCHEMBL6821752 0.82 CA1 (0.45) PTPN1PTPN6PTPN11CA1CA2
SCHEMBL6821033 0.80 PTPN1 (0.46) PTPN1PTPN6PTPN11ALDH1A1NR1I2
SCHEMBL6818212 0.72 PPID (0.41) CA1CA2CA12CA14ALDH1A1
SCHEMBL6824712 0.72 ALDH1A1 (0.47) CA1CA2CA12CA14ALDH1A1
SCHEMBL5120240 0.69 CA12 (0.40) PTPN1PTPN6PTPN11CA1CA2
SCHEMBL5892950 0.69 ITGB3 (0.46) PTPN1CYP2C9CYP2C19HTT
SCHEMBL1731086 0.69 GAA (0.46) CA1CA2CA12CA14ALDH1A1
SCHEMBL15354550 0.67 CA12 (0.39) CA1CA2CA12CA14ALDH1A1
SCHEMBL14805406 0.67 NR1H2 (0.41) PTPN1PTPN6PTPN11NR1H2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004050646-A1 1, 2, 5-THIADIAZOLIDIN-3-ONE 1, 1 DIOXIDE DERIVATIVES AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE PTP1B ASTRAZENECA AB (SE) 2004-06-17 WO disclosed