SCHEMBL6822002

SCHEMBL6822002

COc1cc(CNC(C)=O)ccc1[N+](=O)[O-]

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C19 P33261 1/20 0.51
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
MAPT P10636 1/20 0.48
PDE7A Q13946 1/20 0.47
PDE3A Q14432 1/20 0.47
ATM Q13315 1/20 0.47
NQO2 P16083 1/20 0.47
MTNR1A P48039 1/20 0.47
MTNR1B P49286 1/20 0.47
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5312469 0.89 ALDH1A1 (0.52) ALDH1A1CYP1A2CYP3A4CYP2C19MEN1
SCHEMBL5718757 0.83 ALDH1A1 (0.47) ALDH1A1CYP1A2CYP3A4CYP2C19MEN1
SCHEMBL25734367 0.81 ALDH1A1 (0.49) ALDH1A1CYP1A2CYP3A4CYP2C19MEN1
SCHEMBL6171639 0.81 ALDH1A1 (0.78) ALDH1A1MEN1KMT2A
SCHEMBL2593349 0.80 CYP1A2 (0.50) ALDH1A1CYP1A2CYP3A4CYP2C19MEN1
SCHEMBL29750606 0.79 TTR (0.64) ALDH1A1CYP1A2CYP3A4CYP2C19MEN1
SCHEMBL704754 0.79 TTR (0.64) ALDH1A1CYP1A2CYP3A4CYP2C19MEN1
SCHEMBL30286022 0.78 POLB (0.49) ALDH1A1MEN1KMT2AMAPTHPGD
SCHEMBL2593397 0.78 ALDH1A1 (0.60) ALDH1A1CYP1A2CYP3A4CYP2C19MAPT
SCHEMBL5673785 0.78 ALDH1A1 (0.60) ALDH1A1CYP1A2CYP3A4CYP2C19MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004050646-A1 1, 2, 5-THIADIAZOLIDIN-3-ONE 1, 1 DIOXIDE DERIVATIVES AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE PTP1B ASTRAZENECA AB (SE) 2004-06-17 WO disclosed